SCHEMBL2836044

SCHEMBL2836044

Cc1cc2c(o1)CN(C)CC2Oc1ccc(C(F)(F)F)cc1

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 5/20 0.36
HRH3 Q9Y5N1 3/20 0.36
MCHR1 Q99705 6/20 0.34
SLC6A2 P23975 2/20 0.34
FPR2 P25090 1/20 0.33
PROKR1 Q8TCW9 1/20 0.33
CCR6 P51684 1/20 0.32
KCNH2 Q12809 1/20 0.32
PTGS2 P35354 1/20 0.32
LIPG Q9Y5X9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2838582 0.88 MCHR1 (0.39) SLC6A4HRH3MCHR1FPR2PROKR1
Hydrochloric Acid SCHEMBL2836932 0.83 SLC6A4 (0.36) SLC6A4HRH3SLC6A2
Hydrochloric Acid SCHEMBL2835799 0.79 SLC9A3 (0.38) SLC6A4HRH3PTGS2
Hydrochloric Acid SCHEMBL2839559 0.79 SLC6A4 (0.36) SLC6A4HRH3SLC6A2FPR2PROKR1
Hydrochloric Acid SCHEMBL3580232 0.79 SLC6A2 (0.31) SLC6A4SLC6A2
Hydrochloric Acid SCHEMBL2841523 0.79 SLC6A2 (0.38) SLC6A4HRH3SLC6A2FPR2PROKR1
Hydrochloric Acid SCHEMBL2835058 0.76 AR (0.34)
Hydrochloric Acid SCHEMBL3579144 0.76 MCHR1 (0.33) MCHR1
Hydrochloric Acid SCHEMBL2844337 0.76
Hydrochloric Acid SCHEMBL2837907 0.76 SMN1; SMN2 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8217031-B2 Heteroaryl derivatives NIPPON SHINYAKU CO., LTD. (JP) 2012-07-10 US disclosed
US-20100048537-A1 HETEROARYL DERIVATIVES NIPPON SHINYAKU CO., LTD. (JP) 2010-02-25 US disclosed
EP-2141168-A1 HETEROARYL DERIVATIVES Nippon Shinyaku Co., Ltd. (JP) 2010-01-06 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100048537-A1 HETEROARYL DERIVATIVES OPRD1, OPRM1, OPRK1 SLC6A4 185/4885HRH3 777/4885MCHR1 401/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.