SCHEMBL28362008

SCHEMBL28362008

COc1ccc(Cc2ccnc(N)c2C)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.50
CYP2D6 P10635 1/20 0.50
ATM Q13315 1/20 0.50
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
POLB P06746 1/20 0.47
MPO P05164 1/20 0.46
ROCK1 Q13464 2/20 0.45
LMNA P02545 2/20 0.44
HPGD P15428 1/20 0.44
DHFR P00374 1/20 0.44
NPSR1 Q6W5P4 1/20 0.43
LTA4H P09960 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
PDE3B Q13370 1/20 0.43
PDE3A Q14432 1/20 0.43
PDE10A Q9Y233 1/20 0.43
IDO1 P14902 1/20 0.42
NOS3 P29474 1/20 0.42
NOS2 P35228 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9535888 0.86 ALDH1A1 (0.51) ALDH1A1CYP2D6ATMNPC1RAB9A
SCHEMBL23045757 0.84 ALDH1A1 (0.58) ALDH1A1CYP2D6ATMNPC1RAB9A
Ammonia Solution, Strong SCHEMBL25279198 0.83 ALDH1A1 (0.56) ALDH1A1CYP2D6ATMNPC1RAB9A
Ammonia Solution, Strong SCHEMBL28361999 0.81 PDE3B (0.52) ALDH1A1CYP2D6ATMNPC1RAB9A
SCHEMBL9391619 0.79 NPC1 (0.61) ALDH1A1CYP2D6ATMNPC1RAB9A
SCHEMBL31279567 0.79 MPO (0.47) ALDH1A1CYP2D6ATMNPC1RAB9A
SCHEMBL29937376 0.77 ALDH1A1 (0.56) ALDH1A1CYP2D6ATMPOLBLMNA
Ammonia Solution, Strong SCHEMBL2450875 0.77 ALDH1A1 (0.53) ALDH1A1CYP2D6ATMNPC1RAB9A
SCHEMBL3551608 0.77 NPC1 (0.67) ALDH1A1CYP2D6ATMNPC1RAB9A
SCHEMBL28522308 0.76 ALDH1A1 (0.51) ALDH1A1CYP2D6ATMNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117024411-A Isoquinoline as HPK1 inhibitor 豪夫迈·罗氏有限公司 2023-11-10 CN disclosed
CN-110709392-B Isoquinoline as HPK1 inhibitor 豪夫迈·罗氏有限公司 2023-09-29 CN disclosed
CN-110709392-A Isoquinoline as HPK1 inhibitors 豪夫迈·罗氏有限公司 2020-01-17 CN disclosed