SCHEMBL29937376

SCHEMBL29937376

COc1ccc(Cc2cnc(N)c(Cc3ccc(OC)cc3)c2C)cc1

nearest known ligand 0.62

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.56
CYP2D6 P10635 1/20 0.56
ATM Q13315 1/20 0.56
NPSR1 Q6W5P4 1/20 0.49
LMNA P02545 2/20 0.49
POLB P06746 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
DHFR P00374 4/20 0.47
CSF1R P07333 2/20 0.46
NTRK2 Q16620 2/20 0.46
NTRK1 P04629 1/20 0.46
NTRK3 Q16288 1/20 0.46
PKM P14618 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30998660 0.88 ALDH1A1 (0.48) ALDH1A1CYP2D6ATMNPSR1LMNA
SCHEMBL28996034 0.88 ALDH1A1 (0.56) ALDH1A1CYP2D6ATMNPSR1LMNA
SCHEMBL29687392 0.88 ALDH1A1 (0.56) ALDH1A1CYP2D6ATMNPSR1LMNA
SCHEMBL28515732 0.82 ALDH1A1 (0.50) ALDH1A1CYP2D6ATMNPSR1LMNA
SCHEMBL23045757 0.80 ALDH1A1 (0.58) ALDH1A1CYP2D6ATMNPSR1LMNA
SCHEMBL29433996 0.80 ALDH1A1 (0.58) ALDH1A1CYP2D6ATMNPSR1LMNA
SCHEMBL28729752 0.80 ALDH1A1 (0.58) ALDH1A1CYP2D6ATMNPSR1LMNA
Ammonia Solution, Strong SCHEMBL25279198 0.79 ALDH1A1 (0.56) ALDH1A1CYP2D6ATMNPSR1LMNA
SCHEMBL28039300 0.79 DHFR (0.57) ALDH1A1CYP2D6ATMLMNADHFR
Hydrochloric Acid SCHEMBL7522555 0.78 ALDH1A1 (0.68) ALDH1A1CYP2D6ATMNPSR1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4499639-A1 HETEROCYCLIC COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH BeiGene, Ltd. (KY) 2025-02-05 EP disclosed
CN-118900838-A Heterocyclic compounds, compositions thereof and methods of treatment thereof 百济神州有限公司 2024-11-05 CN disclosed
EP-4322954-A1 SMALL MOLECULE INHIBITORS OF KRAS G12D MUTANT Merck Sharp & Dohme LLC (US) 2024-02-21 EP disclosed
CN-117242074-A KRAS G12D inhibitors 百时美施贵宝公司 2023-12-15 CN disclosed
WO-2023179703-A1 HETEROCYCLIC COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH BEIGENE , LTD. (KY) 2023-09-28 WO disclosed
WO-2022221739-A1 SMALL MOLECULE INHIBITORS OF KRAS G12D MUTANT MERCK SHARP & DOHME CORP. (US) 2022-10-20 WO disclosed