SCHEMBL28369459

SCHEMBL28369459

O=C(Cc1c[nH]c2ccccc12)Nc1ccncc1Cl

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GALR3 O60755 1/20 0.57
NR2F2 P24468 1/20 0.57
GLA P06280 1/20 0.56
MAPT P10636 4/20 0.54
MEN1 O00255 2/20 0.54
STAT3 P40763 2/20 0.54
KMT2A Q03164 2/20 0.54
RAB9A P51151 1/20 0.54
HSD17B10 Q99714 1/20 0.54
PKM P14618 2/20 0.54
ALDH1A1 P00352 1/20 0.54
HTT P42858 1/20 0.54
LMNA P02545 3/20 0.53
CCKBR P32239 1/20 0.53
CYP1A2 P05177 1/20 0.51
POLB P06746 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28373298 0.86 GLA (0.56) GLAMAPTMEN1STAT3KMT2A
SCHEMBL28885922 0.86 LMNA (0.57) GLAMAPTMEN1STAT3KMT2A
SCHEMBL28373392 0.85 MAPT (0.59) GLAMAPTMEN1STAT3KMT2A
SCHEMBL28374001 0.80 GLA (0.62) GLAMAPTMEN1STAT3KMT2A
SCHEMBL28167913 0.80 ALDH1A1 (0.64) GLAMAPTMEN1STAT3KMT2A
SCHEMBL28369453 0.77 MAPT (0.58) GLAMAPTMEN1STAT3KMT2A
SCHEMBL28369557 0.76 MAPT (0.58) GLAMAPTMEN1STAT3KMT2A
SCHEMBL12845374 0.76 HRH3 (0.60) GLAMAPTMEN1STAT3KMT2A
SCHEMBL28369958 0.76 GALR3 (0.56) GALR3NR2F2MAPTALDH1A1HTT
SCHEMBL18229447 0.75 MAPT (0.57) GLAMAPTMEN1STAT3KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107149602-B Application of indole compounds and derivatives thereof in preparation of anti-HIV drugs 中国医学科学院药物研究所 2020-10-09 CN disclosed
CN-107149603-B Application of indole compounds and derivatives thereof in preparation of anti-influenza virus drugs 中国医学科学院药物研究所 2020-07-14 CN disclosed
CN-107176921-B Indole compounds with antiviral activity in isatis root and derivatives thereof 中国医学科学院药物研究所 2020-03-31 CN disclosed