SCHEMBL28375002

SCHEMBL28375002

COc1ccc(-n2nc(S)nc2-c2cc(OC)c(OC)c(OC)c2)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 6/20 0.63
PTGS1 P23219 4/20 0.51
HDAC4 P56524 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
LMNA P02545 2/20 0.44
USP2 O75604 1/20 0.44
ALDH1A1 P00352 1/20 0.44
HPGD P15428 1/20 0.44
TSHR P16473 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HSD17B10 Q99714 1/20 0.44
MEN1 O00255 1/20 0.43
GAA P10253 1/20 0.43
KMT2A Q03164 1/20 0.43
APOBEC3G Q9HC16 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
MAP3K11 Q16584 1/20 0.42
TP53 P04637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28371151 0.88 PTGS2 (0.50) PTGS2HDAC4HDAC1HDAC2HDAC6
SCHEMBL28371338 0.88 PTGS2 (0.53) PTGS2HDAC4HDAC1HDAC2HDAC6
SCHEMBL28886199 0.88 PTGS2 (0.50) PTGS2HDAC4HDAC1HDAC2HDAC6
SCHEMBL28376412 0.88 PTGS2 (0.50) PTGS2HDAC4HDAC1HDAC2HDAC6
SCHEMBL6132166 0.84 PTGS2 (0.69) PTGS2PTGS1LMNAHPGDSMN1; SMN2
SCHEMBL11376435 0.81 L3MBTL1 (0.62) PTGS2PTGS1ALDH1A1HPGDSMN1; SMN2
SCHEMBL28198327 0.78 PTGS2 (0.56) PTGS2PTGS1LMNAUSP2ALDH1A1
SCHEMBL11376339 0.75 PTGS1 (0.51) PTGS2PTGS1LMNAALDH1A1SMN1; SMN2
SCHEMBL11318935 0.75 PTGS2 (0.52) PTGS2HDAC4HDAC1HDAC2HDAC6
SCHEMBL28233689 0.72 LMNA (0.57) PTGS2PTGS1LMNAALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104910082-B 3,4, 5-trisubstituted-1, 2, 4-triazole thioether derivative and synthesis method and application thereof 贵阳学院 2020-03-17 CN disclosed