SCHEMBL28375035

SCHEMBL28375035

COC(=O)c1ccc2c(ccn2-c2ncccn2)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 1/20 0.55
HTT P42858 1/20 0.55
FGFR1 P11362 2/20 0.48
KDM4E B2RXH2 4/20 0.43
CYP19A1 P11511 1/20 0.43
CYP11B1 P15538 1/20 0.43
CYP11B2 P19099 1/20 0.43
JMJD6 Q6NYC1 1/20 0.42
MGLL Q99685 2/20 0.41
ROCK1 Q13464 2/20 0.41
POLB P06746 3/20 0.41
GAA P10253 1/20 0.41
TSHR P16473 1/20 0.41
KDM6B O15054 1/20 0.40
KDM5C P41229 1/20 0.40
KDM4C Q9H3R0 1/20 0.40
KDM2A Q9Y2K7 1/20 0.40
KDM3A Q9Y4C1 1/20 0.40
ROCK2 O75116 1/20 0.40
PIM1 P11309 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3973189 0.86 POLB (0.55) ALOX15HTTFGFR1KDM4ECYP19A1
SCHEMBL31556376 0.86 POLB (0.55) ALOX15HTTFGFR1KDM4ECYP19A1
SCHEMBL2610310 0.83 POLB (0.48) FGFR1KDM4EMGLLROCK1POLB
SCHEMBL3975054 0.81 FGFR1 (0.60) ALOX15HTTFGFR1KDM4EMGLL
SCHEMBL31525708 0.80 HTT (0.48) ALOX15HTTFGFR1KDM4ECYP19A1
SCHEMBL31525861 0.80 ALOX15 (0.47) ALOX15HTTFGFR1KDM4ECYP19A1
SCHEMBL31525835 0.80 ALDH1A1 (0.54) ALOX15HTTFGFR1KDM4ECYP19A1
SCHEMBL958825 0.79 ROCK1 (0.47) ALOX15HTTFGFR1KDM4EJMJD6
SCHEMBL28312597 0.77 RXRA (0.46) ALOX15HTTFGFR1KDM4EPOLB
SCHEMBL28674784 0.77 MAPT (0.46) ALOX15HTTFGFR1KDM4ECYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112574180-B N-2-pyrimidinyl-3-fluoroindole compound and preparation method and application thereof 浙江工业大学 2021-10-15 CN disclosed
CN-112574180-A N-2-pyrimidinyl-3-fluoroindole compound and preparation method and application thereof 浙江工业大学 2021-03-30 CN disclosed
CN-106279236-B Method for synthesizing 2-triisopropyl silicon-based acetylene indole compound 南京理工大学 2020-04-10 CN disclosed