SCHEMBL28375403

SCHEMBL28375403

O=C(O)c1ccc(-c2cnn(C3CCCCO3)c2)nc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.45
LDHA P00338 2/20 0.44
P4HA1 P13674 2/20 0.42
P4HTM Q9NXG6 1/20 0.42
KDM5B Q9UGL1 1/20 0.42
CYP4F2 P78329 1/20 0.41
CYP4A11 Q02928 1/20 0.41
HCAR3 P49019 3/20 0.41
FGFR1 P11362 2/20 0.41
FLT3 P36888 2/20 0.41
FGFR2 P21802 1/20 0.41
FGFR4 P22455 1/20 0.41
FGFR3 P22607 1/20 0.41
KDR P35968 1/20 0.41
OXTR P30559 2/20 0.39
AVPR1A P37288 2/20 0.39
USP30 Q70CQ3 1/20 0.38
CD274 Q9NZQ7 1/20 0.38
RXRA P19793 1/20 0.38
RXRB P28702 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23535740 0.86 MCL1 (0.47) MCL1KDM5BCYP4F2CYP4A11HCAR3
SCHEMBL19277419 0.83 CYP4F2 (0.43) MCL1KDM5BCYP4F2CYP4A11FGFR1
SCHEMBL29689591 0.83 KDM5B (0.44) MCL1KDM5BCYP4F2CYP4A11FGFR1
SCHEMBL29218244 0.81 KDM5B (0.42) MCL1KDM5BCYP4F2CYP4A11FGFR1
SCHEMBL30895651 0.81 KDM5B (0.42) MCL1KDM5BCYP4F2CYP4A11FGFR1
SCHEMBL26130683 0.81 KDM5B (0.42) MCL1KDM5BCYP4F2CYP4A11FGFR1
SCHEMBL31434739 0.81 FLT3 (0.45) MCL1KDM5BCYP4F2CYP4A11FGFR1
Fluoride SCHEMBL14796503 0.80 ACHE (0.43) MCL1KDM5BCYP4F2CYP4A11HCAR3
SCHEMBL5139638 0.80 ACHE (0.43) MCL1KDM5BCYP4F2CYP4A11HCAR3
SCHEMBL16896639 0.79 CYP4F2 (0.48) MCL1KDM5BCYP4F2CYP4A11FGFR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111362966-B Bicyclic heterocyclic derivatives as IRAK4 inhibitors 奥列基因发现技术有限公司 2022-03-11 CN disclosed
CN-111362966-A Bicyclic heterocyclic derivatives as IRAK4 inhibitors 奥列基因发现技术有限公司 2020-07-03 CN disclosed
CN-106456619-B Bicyclic heterocyclic derivatives as IRAK4 inhibitors 奥列基因发现技术有限公司 2020-03-27 CN disclosed