SCHEMBL28378128

SCHEMBL28378128

CCCc1nn(C)c2c(Nc3cccc(C(F)(F)F)c3)nc(/C=C/c3ccccc3)nc12

nearest known ligand 0.62

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.41
MAPT P10636 1/20 0.41
IDH2 P48735 1/20 0.39
BCDIN3D Q7Z5W3 3/20 0.38
NPY1R P25929 1/20 0.38
NPY5R Q15761 1/20 0.38
ABCG2 Q9UNQ0 2/20 0.38
KDR P35968 1/20 0.37
EGFR P00533 1/20 0.37
CTSC P53634 1/20 0.37
PDE5A O76074 1/20 0.37
TSHR P16473 1/20 0.37
HTT P42858 1/20 0.37
FYN P06241 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28378129 1.00 TP53 (0.41) TP53MAPTIDH2BCDIN3DNPY1R
SCHEMBL28373456 0.88 TERT (0.51) TP53MAPTABCG2EGFRHTT
SCHEMBL28373459 0.88 TERT (0.51) TP53MAPTABCG2EGFRHTT
SCHEMBL28373321 0.82 PTGS2 (0.42) PDE5A
SCHEMBL28373320 0.82 PTGS2 (0.42) PDE5A
SCHEMBL28375715 0.81 PDE5A (0.39) BCDIN3DPDE5A
Hydrochloric Acid SCHEMBL5356288 0.79 ABCG2 (0.47) TP53MAPTBCDIN3DABCG2CTSC
SCHEMBL28375718 0.78 TERT (0.57) EGFR
SCHEMBL28375719 0.78 TERT (0.57) EGFR
SCHEMBL28374607 0.77 PDE5A (0.43) PDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108503648-B Styryl pyrazolopyrimidine compound, pharmaceutical composition, preparation method and application 安徽医科大学 2020-04-14 CN disclosed