SCHEMBL2838918

SCHEMBL2838918

CC(=O)N(c1ccccc1)c1cc(CN(C)C(=O)O)nn1-c1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.37
GRM5 P41594 1/20 0.37
ALDH1A1 P00352 4/20 0.37
LMNA P02545 2/20 0.37
TSHR P16473 2/20 0.35
POLB P06746 2/20 0.35
MAPK1 P28482 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
CRHBP P24387 1/20 0.35
CRHR2 Q13324 1/20 0.35
MTNR1A P48039 1/20 0.34
MTNR1B P49286 1/20 0.34
NPC1 O15118 1/20 0.34
XBP1 P17861 1/20 0.34
HTT P42858 1/20 0.34
RAB9A P51151 1/20 0.34
PAX8 Q06710 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
SLC16A3 O15427 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2838656 0.86 ALDH1A1 (0.39) NPSR1GRM5ALDH1A1LMNATSHR
SCHEMBL3012799 0.86 HTR2C (0.49) NPSR1GRM5ALDH1A1LMNATSHR
SCHEMBL3012801 0.83 ALDH1A1 (0.34) NPSR1GRM5ALDH1A1LMNATSHR
SCHEMBL2836798 0.82 MEN1 (0.39) NPSR1ALDH1A1LMNATSHRPOLB
SCHEMBL2838922 0.80 ALDH1A1 (0.43) NPSR1ALDH1A1LMNATSHRPOLB
SCHEMBL18093107 0.77 CA1 (0.41) NPSR1ALDH1A1LMNAPOLBGAA
SCHEMBL3012796 0.75 RIPK1 (0.38) ALDH1A1MAPK1
SCHEMBL2840465 0.73 GAA (0.53) ALDH1A1LMNATSHRMAPK1HTT
SCHEMBL2833994 0.73 HTR2C (0.52) ALDH1A1LMNASLC16A3SLC16A1CNR1
SCHEMBL19181130 0.68 BCL2 (0.43) NPSR1ALDH1A1TSHRKMT2AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3162798-A1 5-MEMBERED HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2017-05-03 EP disclosed
EP-2196459-B1 5-MEMBERED HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICAL (JP) 2016-11-02 EP disclosed
EP-2196459-A1 5-MEMBERED HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2010-06-16 EP disclosed