SCHEMBL28392020

SCHEMBL28392020

Fc1ccc2ccnc(Cl)c2c1.O=c1[nH]ccc2ccc(F)cc12

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.43
CHEK1 O14757 2/20 0.42
JAK2 O60674 11/20 0.40
AHR P35869 1/20 0.39
TYMS P04818 2/20 0.38
JAK1 P23458 1/20 0.38
TYK2 P29597 1/20 0.38
JAK3 P52333 1/20 0.38
ROCK2 O75116 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5983565 0.86 JAK2 (0.41) PARP1CHEK1JAK2AHRTYMS
SCHEMBL26071728 0.85 ROCK2 (0.44) PARP1CHEK1ROCK2
SCHEMBL30596156 0.85 ROCK2 (0.44) PARP1CHEK1ROCK2
SCHEMBL30673402 0.83 PARP1 (0.53) PARP1CHEK1JAK2AHRTYMS
SCHEMBL1536413 0.83 PARP1 (0.53) PARP1CHEK1JAK2AHRTYMS
SCHEMBL1315422 0.83 MAPT (0.47) TYMS
SCHEMBL28397791 0.77 PARP1 (0.66) PARP1CHEK1JAK2JAK3
SCHEMBL21870525 0.72 MAPT (0.61) TYMS
Trifluoromethanesulfonic Acid SCHEMBL27781740 0.71 PARP1 (0.42) PARP1CHEK1JAK2AHRTYMS
SCHEMBL722687 0.71 MAPT (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111138355-A Preparation method of formaldehyde-substituted aza-condensed ring compound 成都睿智化学研究有限公司 2020-05-12 CN disclosed