SCHEMBL28396299

SCHEMBL28396299

OC1(c2cncc3ccccc23)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 12/20 0.43
CYP11B1 P15538 11/20 0.43
PRKCZ Q05513 1/20 0.39
ADRA2A P08913 1/20 0.38
ADRA2B P18089 1/20 0.38
ADRA2C P18825 1/20 0.38
ADRA1A P35348 1/20 0.38
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37
SLC6A3 Q01959 1/20 0.37
KDM4E B2RXH2 2/20 0.35
MAPKAPK2 P49137 1/20 0.35
CYP17A1 P05093 1/20 0.35
CYP3A4 P08684 1/20 0.35
GPR3 P46089 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2B6 P20813 1/20 0.34
CYP2C19 P33261 1/20 0.34
ITGA4 P13612 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7964139 0.89 CYP11B1 (0.46) CYP11B2CYP11B1PRKCZADRA2AADRA2B
SCHEMBL30344013 0.78 CYP11B1 (0.43) CYP11B2CYP11B1PRKCZADRA2AADRA2B
SCHEMBL28033596 0.78 CYP11B2 (0.43) CYP11B2CYP11B1PRKCZADRA2AADRA2B
SCHEMBL25155485 0.78 CYP11B1 (0.43) CYP11B2CYP11B1PRKCZADRA2AADRA2B
SCHEMBL29874979 0.78 CYP11B1 (0.43) CYP11B2CYP11B1PRKCZADRA2AADRA2B
SCHEMBL7964475 0.76 CYP11B2 (0.41) CYP11B2CYP11B1ITGA4ITGB7
SCHEMBL28485903 0.76 SLC6A3 (0.49) SLC6A2SLC6A4SLC6A3KDM4ECYP3A4
SCHEMBL28389056 0.75 CYP11B1 (0.41) CYP11B2CYP11B1PRKCZADRA2AADRA2B
SCHEMBL31513789 0.69 SLC6A3 (0.54) SLC6A2SLC6A4SLC6A3KDM4ECYP3A4
SCHEMBL30344744 0.69 SLC6A3 (0.50) SLC6A2SLC6A4SLC6A3KDM4ECYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111116555-B Rho kinase inhibitor and preparation method and application thereof 北京盈科瑞创新药物研究有限公司 2023-06-02 CN disclosed
CN-111116555-A Rho kinase inhibitor and preparation method and application thereof 北京盈科瑞创新药物研究有限公司 2020-05-08 CN disclosed