SCHEMBL28396337

SCHEMBL28396337

O=C1CCN(C(=O)c2ccc(Br)cc2)C1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.61
CA12 O43570 1/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
CA7 P43166 1/20 0.50
CA9 Q16790 1/20 0.50
CA14 Q9ULX7 1/20 0.50
POLB P06746 1/20 0.50
L3MBTL3 Q96JM7 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
LMNA P02545 1/20 0.47
ABL1 P00519 2/20 0.46
BCR P11274 2/20 0.46
GPR183 P32249 1/20 0.46
MGLL Q99685 1/20 0.46
HSD11B1 P28845 1/20 0.46
HSP90AA1 P07900 1/20 0.44
ALDH1A1 P00352 1/20 0.44
MTHFD2 P13995 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26987208 0.89 HPGD (0.70) HPGDCA12CA1CA2CA7
Ethylene SCHEMBL8378361 0.86 HPGD (0.66) HPGDCA12CA1CA2CA7
SCHEMBL694171 0.85 HPGD (0.63) HPGDCA12CA1CA2CA7
SCHEMBL6558877 0.83 CA1 (0.51) HPGDCA12CA1CA2CA7
SCHEMBL7469385 0.82 HPGD (0.56) HPGDLMNAALDH1A1MTHFD2
SCHEMBL7047272 0.80 HPGD (0.63) HPGDPOLBLMNAALDH1A1KMT2A
SCHEMBL24120195 0.79 HPGD (0.61) HPGDPOLBL3MBTL3L3MBTL1LMNA
SCHEMBL7380773 0.79 ALDH1A1 (0.52) CA1CA2L3MBTL1GPR183ALDH1A1
SCHEMBL644199 0.76 HPGD (0.92) HPGDCA12CA1CA2CA7
SCHEMBL971083 0.76 HPGD (1.00) HPGDCA12CA1CA2CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111116585-B Compound with c-MET kinase inhibitory activity, preparation method, composition and application 北京鑫开元医药科技有限公司 2021-02-05 CN disclosed
CN-111116585-A Compound with c-MET kinase inhibitory activity, preparation method, composition and application 北京鑫开元医药科技有限公司 2020-05-08 CN disclosed