SCHEMBL7380773

SCHEMBL7380773

N#Cc1ccc(C(=O)N2CCC(=O)C2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.52
PDK1 Q15118 1/20 0.49
PDK2 Q15119 1/20 0.49
PDK3 Q15120 1/20 0.49
PDK4 Q16654 1/20 0.49
SLC6A7 Q99884 1/20 0.48
EPHX2 P34913 1/20 0.46
GPR183 P32249 1/20 0.46
MAPT P10636 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
NAMPT P43490 2/20 0.44
HRH3 Q9Y5N1 3/20 0.43
CYP2D6 P10635 2/20 0.43
HRH1 P35367 1/20 0.43
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
KCNA5 P22460 1/20 0.43
GRM5 P41594 1/20 0.43
KCNH2 Q12809 1/20 0.42
PRLHR P49683 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7828410 0.90 ALDH1A1 (0.55) ALDH1A1PDK1PDK2PDK3PDK4
Ethylene SCHEMBL7964704 0.88 ALDH1A1 (0.52) ALDH1A1PDK1PDK2PDK3PDK4
SCHEMBL6558877 0.79 CA1 (0.51) ALDH1A1CA1CA2
SCHEMBL28396337 0.79 HPGD (0.61) ALDH1A1GPR183L3MBTL1CA1CA2
SCHEMBL8103530 0.79 CA1 (0.64) ALDH1A1MAPTNAMPTCA1CA2
SCHEMBL31387924 0.78 HPGD (0.68) ALDH1A1PDK1PDK2PDK3PDK4
SCHEMBL7469385 0.78 HPGD (0.56) ALDH1A1
SCHEMBL31387922 0.78 HPGD (0.68) ALDH1A1PDK1PDK2PDK3PDK4
SCHEMBL3633068 0.77 HPGD (0.71) ALDH1A1PDK1PDK2PDK3PDK4
SCHEMBL7047272 0.76 HPGD (0.63) ALDH1A1SLC6A7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0936912-A4 INHIBITORS OF CYSTEINE PROTEASE SMITHKLINE BEECHAM CORP (US) 1999-10-13 EP disclosed
EP-0936912-A1 INHIBITORS OF CYSTEINE PROTEASE SMITHKLINE BEECHAM CORPORATION (US) 1999-08-25 EP disclosed
WO-1998005336-A1 INHIBITORS OF CYSTEINE PROTEASE SMITHKLINE BEECHAM CORPORATION (US) 1998-02-12 WO disclosed