SCHEMBL28396455

SCHEMBL28396455

FC(F)(F)c1[c]cccc1COCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.47
TACR1 P25103 4/20 0.43
CES1 P23141 1/20 0.35
KDM4E B2RXH2 3/20 0.35
POLB P06746 2/20 0.35
CA1 P00915 1/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
ALDH1A1 P00352 2/20 0.33
NPC1 O15118 1/20 0.33
LMNA P02545 1/20 0.33
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33
MAPK1 P28482 1/20 0.33
HTT P42858 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
IDO1 P14902 1/20 0.33
CACNA1F O60840 1/20 0.33
CACNA1D Q01668 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8939764 0.80 HTR2A (0.39) CES1KDM4EALDH1A1SMN1; SMN2
SCHEMBL27602767 0.79 MAOB (0.42) KDM4ESMN1; SMN2
SCHEMBL4280049 0.76 MAPT (0.46) L3MBTL1NPC1MAPTMAPK1TDP1
SCHEMBL27584915 0.75 POLB (0.35) CES1KDM4EPOLBALDH1A1NPC1
SCHEMBL7423138 0.72 TSHR (0.47) TSHRTACR1KDM4EPOLBCA1
SCHEMBL7425373 0.72 TSHR (0.47) TSHRTACR1KDM4EPOLBCA1
SCHEMBL7401991 0.71 GABRA1 (0.40) CACNA1C
SCHEMBL17046318 0.71 PDK2 (0.33)
SCHEMBL27937767 0.71
SCHEMBL27899133 0.71 PNMT (0.34) IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107001332-B Piperidine derivatives 豪夫迈·罗氏有限公司 2020-05-15 CN disclosed