SCHEMBL28397669

SCHEMBL28397669

CCOC(=O)c1nc(CNC(=O)O)sc1Br

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
ALDH1A1 P00352 4/20 0.42
CYP1A2 P05177 2/20 0.42
GAA P10253 2/20 0.41
TRPM8 Q7Z2W7 1/20 0.39
MAPT P10636 3/20 0.38
RAB9A P51151 2/20 0.38
LMNA P02545 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
KDM4E B2RXH2 2/20 0.37
NPSR1 Q6W5P4 2/20 0.37
DHODH Q02127 1/20 0.37
HPGD P15428 3/20 0.37
TSHR P16473 1/20 0.37
TARBP2 Q15633 1/20 0.36
ILK Q13418 1/20 0.36
NPC1 O15118 1/20 0.36
CDC7 O00311 1/20 0.36
DBF4 Q9UBU7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28392396 0.88 NPSR1 (0.40) MEN1KMT2AALDH1A1GAATRPM8
SCHEMBL28959134 0.85 MEN1 (0.53) MEN1KMT2AALDH1A1CYP1A2GAA
SCHEMBL20743931 0.83 MEN1 (0.46) MEN1KMT2AALDH1A1CYP1A2GAA
SCHEMBL5731466 0.83 ALDH1A1 (0.47) MEN1KMT2AALDH1A1CYP1A2GAA
SCHEMBL28397631 0.83 MEN1 (0.42) MEN1KMT2AALDH1A1CYP1A2GAA
SCHEMBL28397369 0.83 L3MBTL1 (0.43) MEN1KMT2AALDH1A1CYP1A2GAA
SCHEMBL10317436 0.82 ALDH1A1 (0.46) MEN1KMT2AALDH1A1CYP1A2GAA
SCHEMBL12850213 0.81 MEN1 (0.45) MEN1KMT2AALDH1A1CYP1A2GAA
SCHEMBL18781580 0.81 MEN1 (0.45) MEN1KMT2AALDH1A1CYP1A2GAA
SCHEMBL28395679 0.81 MEN1 (0.41) MEN1KMT2AALDH1A1CYP1A2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110997682-A Inhibitors of indoleamine 2, 3-dioxygenase and/or tryptophan 2, 3-dioxygenase 爱杜西亚药品有限公司 2020-04-10 CN disclosed