SCHEMBL28400595

SCHEMBL28400595

COC1OC(=O)C(Br)=C1Br

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NUAK1 O60285 1/20 0.38
IGF1R P08069 1/20 0.38
MET P08581 1/20 0.38
SRC P12931 1/20 0.38
AXL P30530 1/20 0.38
KDR P35968 1/20 0.38
NEK2 P51955 1/20 0.38
PTK2 Q05397 1/20 0.38
AURKB Q96GD4 1/20 0.38
ALK Q9UM73 1/20 0.38
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29822164 0.77 KMT2A (0.37)
SCHEMBL28393133 0.77 ALDH1A1 (0.38)
SCHEMBL30104877 0.77 NUAK1 (0.35) NUAK1IGF1RMETSRCAXL
SCHEMBL30104878 0.72 NUAK1 (0.33) NUAK1IGF1RMETSRCAXL
SCHEMBL29822002 0.71 KDM4E (0.35) KDM4E
SCHEMBL30868879 0.70
SCHEMBL29822108 0.70 CTSV (0.36)
SCHEMBL30104883 0.69 NUAK1 (0.30) NUAK1IGF1RMETSRCAXL
SCHEMBL29822026 0.69 CYP3A4 (0.31)
SCHEMBL16447266 0.64 KDM4E (0.43) NUAK1IGF1RMETSRCAXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115583927-B Thioether compound, and preparation method and application thereof 华南师范大学 2024-07-12 CN disclosed
CN-115583927-A Thioether compound and preparation method and application thereof 华南师范大学 2023-01-10 CN disclosed
CN-109320505-B Preparation and application of halogenated butenolide compound with insecticidal activity 海利尔药业集团股份有限公司 2022-08-02 CN disclosed
CN-109651310-B N-furanone aryl sulfonyl hydrazide derivative and preparation method and application thereof 华南师范大学 2022-07-22 CN disclosed
CN-110511197-B N-furanone aryl sulfonyl hydrazone compound and synthetic method and application thereof 华南师范大学 2021-03-23 CN disclosed
CN-108558797-B Fluorine-containing derivative of bisetherified furanone, preparation method thereof and application of fluorine-containing derivative in preparation of antitumor drugs 华南师范大学 2020-04-17 CN disclosed