SCHEMBL28405063

SCHEMBL28405063

COc1ccc2c(=O)c3ccc(Cl)cc3[nH]c2c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 1/20 0.56
KDM4E B2RXH2 4/20 0.55
CDK4 P11802 2/20 0.52
CCND1 P24385 2/20 0.52
ALDH1A1 P00352 4/20 0.51
MAPT P10636 2/20 0.51
SMN1; SMN2 Q16637 2/20 0.50
CA9 Q16790 1/20 0.50
TP53 P04637 1/20 0.50
HPGD P15428 2/20 0.49
LMNA P02545 2/20 0.49
MEN1 O00255 1/20 0.49
TSHR P16473 1/20 0.49
GFER P55789 1/20 0.49
KMT2A Q03164 1/20 0.49
HSD17B10 Q99714 1/20 0.49
DYRK1A Q13627 1/20 0.48
PARP1 P09874 1/20 0.47
FLT3 P36888 2/20 0.47
ROCK2 O75116 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9709251 0.92 ABCG2 (0.68) ABCG2KDM4ECDK4CCND1ALDH1A1
SCHEMBL14543827 0.84 PARP1 (0.62) KDM4ECDK4CCND1ALDH1A1SMN1; SMN2
SCHEMBL28104195 0.82 ABCG2 (0.82) ABCG2KDM4ECDK4CCND1ALDH1A1
SCHEMBL27174159 0.82 MAPT (0.65) KDM4EALDH1A1MAPTHPGDLMNA
SCHEMBL12015108 0.81 PARP1 (0.58) KDM4ECDK4CCND1ALDH1A1SMN1; SMN2
SCHEMBL29586144 0.81 PARP1 (0.58) KDM4ECDK4CCND1ALDH1A1SMN1; SMN2
SCHEMBL2330779 0.78 KDM4E (0.68) ABCG2KDM4ECDK4CCND1ALDH1A1
SCHEMBL29533596 0.78 KDM4E (0.68) ABCG2KDM4ECDK4CCND1ALDH1A1
SCHEMBL13438413 0.78 ACHE (0.53) KDM4EALDH1A1MAPTPARP1CTSV
SCHEMBL14543826 0.78 PARP1 (0.59) KDM4EALDH1A1MAPTSMN1; SMN2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105884686-B 10-substituted acridine-3 (10) -ketone compound, preparation method and application thereof 中国药科大学 2020-06-09 CN disclosed