SCHEMBL2840801

SCHEMBL2840801

CCN1CCc2sccc2C(Oc2ccc(Cl)c(Cl)c2)C1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 1/20 0.39
KDM4E B2RXH2 2/20 0.39
HHAT Q5VTY9 2/20 0.35
CCR2 P41597 1/20 0.35
KCNH2 Q12809 1/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
SIGMAR1 Q99720 1/20 0.34
ALDH1A1 P00352 1/20 0.34
DRD2 P14416 1/20 0.34
DRD3 P35462 1/20 0.34
LHCGR P22888 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2838307 0.88 KDM4E (0.38) KDM4ECCR2KCNH2SLC6A2SLC6A4
Hydrochloric Acid SCHEMBL2837155 0.87 KDM4E (0.37) OPRD1KDM4EKCNH2SLC6A2SLC6A4
SCHEMBL2836992 0.85 KDM4E (0.38) OPRD1KDM4EHHATKCNH2SLC6A2
Hydrochloric Acid SCHEMBL2840931 0.84 OPRD1 (0.38) OPRD1KDM4EHHATKCNH2SLC6A2
SCHEMBL2841690 0.83 OPRD1 (0.40) OPRD1KDM4ESLC6A2SLC6A4SLC6A3
SCHEMBL2843946 0.77 NPC1 (0.42) KDM4EKCNH2SLC6A2SLC6A4SLC6A3
SCHEMBL2840993 0.75 OPRD1 (0.36) OPRD1KCNH2
SCHEMBL2840576 0.75 DRD3 (0.36) HHATKCNH2SLC6A4SIGMAR1ALDH1A1
Hydrochloric Acid SCHEMBL2841695 0.74 SLC6A4 (0.34) KDM4EKCNH2SLC6A2SLC6A4SLC6A3
SCHEMBL2834956 0.74 HHAT (0.38) KDM4EHHATALDH1A1DRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8217031-B2 Heteroaryl derivatives NIPPON SHINYAKU CO., LTD. (JP) 2012-07-10 US disclosed
US-20100048537-A1 HETEROARYL DERIVATIVES NIPPON SHINYAKU CO., LTD. (JP) 2010-02-25 US disclosed
EP-2141168-A1 HETEROARYL DERIVATIVES Nippon Shinyaku Co., Ltd. (JP) 2010-01-06 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100048537-A1 HETEROARYL DERIVATIVES OPRD1, OPRM1, OPRK1 OPRD1 1/4885KDM4E 3292/4885HHAT 986/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.