SCHEMBL2840920

SCHEMBL2840920

Cc1nc(C2CC2)c(Cc2ccc(-c3ccccc3)c(C#N)c2)c(=O)[nH]1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.42
GAA P10253 2/20 0.42
ALDH1A1 P00352 2/20 0.42
GALR3 O60755 1/20 0.42
HPGD P15428 1/20 0.42
CXCR2 P25025 3/20 0.39
CYP19A1 P11511 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
NR3C1 P04150 2/20 0.38
CYP1A2 P05177 1/20 0.38
CCR2 P41597 2/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
FPR1 P21462 1/20 0.38
CYP2C19 P33261 1/20 0.38
XDH P47989 1/20 0.37
AKT1 P31749 2/20 0.36
AKT2 P31751 2/20 0.36
MAPK1 P28482 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1889453 0.90 KDM4E (0.41) KDM4EGAAALDH1A1GALR3HPGD
SCHEMBL4012582 0.85 KDM4E (0.40) KDM4EGAAALDH1A1GALR3HPGD
SCHEMBL27792468 0.85 CYP1A2 (0.45) KDM4EGAAALDH1A1GALR3HPGD
SCHEMBL27771417 0.84 KDM4E (0.44) KDM4EGAAALDH1A1GALR3HPGD
SCHEMBL27792456 0.81 KDM4E (0.41) KDM4EGAAALDH1A1GALR3HPGD
SCHEMBL27771400 0.80 KDM4E (0.41) KDM4EGAAALDH1A1GALR3HPGD
SCHEMBL27792438 0.80 CYP19A1 (0.39) KDM4EGAAALDH1A1CYP19A1CCR2
SCHEMBL27771371 0.79 ACHE (0.38) KDM4EGAAALDH1A1GALR3HPGD
SCHEMBL27771568 0.75 CCR2 (0.37) KDM4EALDH1A1CYP19A1CCR2SMN1; SMN2
SCHEMBL1894707 0.74 KDM4E (0.38) KDM4EGAAALDH1A1GALR3HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2256115-A1 Heteromonocyclic compound and use thereof Takeda Pharmaceutical Company Limited (JP) 2010-12-01 EP disclosed
CN-101589037-A Heteromonocyclic compounds and uses thereof TAKEDA PHARMACEUTICAL (JP) 2009-11-25 CN disclosed