SCHEMBL28182145

SCHEMBL28182145

C/C=C/c1ccc(Nc2ncnc3cc(N4CCNCC4)c(F)cc23)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 13/20 0.51
HDAC3 O15379 3/20 0.42
HDAC1 Q13547 3/20 0.42
HDAC6 Q9UBN7 3/20 0.42
KDR P35968 3/20 0.39
EPHB4 P54760 3/20 0.39
EPHA2 P29317 2/20 0.39
ERBB2 P04626 2/20 0.39
ABCG2 Q9UNQ0 1/20 0.38
RET P07949 2/20 0.38
HDAC4 P56524 2/20 0.38
HDAC7 Q8WUI4 2/20 0.38
HDAC2 Q92769 2/20 0.38
HDAC10 Q969S8 2/20 0.38
HDAC11 Q96DB2 2/20 0.38
HDAC8 Q9BY41 2/20 0.38
HDAC9 Q9UKV0 2/20 0.38
HDAC5 Q9UQL6 2/20 0.38
KIF5B P33176 1/20 0.38
AURKA O14965 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28409239 0.88 EGFR (0.63) EGFRKDREPHB4EPHA2ERBB2
SCHEMBL7475167 0.87 EGFR (0.51) EGFREPHA2
SCHEMBL28181381 0.82 EGFR (0.53) EGFRHDAC3HDAC1HDAC6KDR
SCHEMBL28411490 0.81 EGFR (0.60) EGFRKDREPHB4ERBB2AURKA
SCHEMBL7473037 0.78 SRC (0.49) EGFRKDRERBB2PDGFRB
SCHEMBL28407547 0.77 EGFR (0.49) EGFRHDAC3HDAC1HDAC6EPHA2
SCHEMBL28181388 0.76 EGFR (0.56) EGFRHDAC3HDAC1HDAC6KDR
SCHEMBL28407194 0.75 EGFR (0.42) EGFRERBB2
SCHEMBL28409241 0.75 EPHA2 (0.49) EGFRKDREPHB4EPHA2
SCHEMBL28409415 0.74 EGFR (0.44) EGFRHDAC3HDAC1HDAC6KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107200715-B Quinazoline derivative and application thereof in preparation of antitumor drugs 陕西师范大学 2020-05-29 CN disclosed
CN-107200715-A Quinazoline derivant and its application in antineoplastic is prepared 陕西师范大学 2017-09-26 CN disclosed