SCHEMBL28409256

SCHEMBL28409256

Cc1nccc(C2CCC(NC(=O)OC(C)(C)C)CC2)c1C

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
JAK1 P23458 6/20 0.50
JAK2 O60674 5/20 0.50
TYK2 P29597 1/20 0.50
JAK3 P52333 1/20 0.50
IDO1 P14902 1/20 0.45
KDM1A O60341 1/20 0.45
MAOB P27338 1/20 0.45
PBK Q96KB5 1/20 0.42
EPHX2 P34913 1/20 0.42
CKS1B P61024 1/20 0.41
SKP1 P63208 1/20 0.41
SKP2 Q13309 1/20 0.41
BTK Q06187 5/20 0.41
DRD2 P14416 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28414964 0.79 OPRL1 (0.46) JAK1JAK2TYK2JAK3KDM1A
SCHEMBL30209415 0.79 OPRL1 (0.46) JAK1JAK2TYK2JAK3KDM1A
SCHEMBL21187176 0.77 IDO1 (0.60) IDO1
SCHEMBL23061556 0.75 IDO1 (0.50) IDO1
SCHEMBL20500390 0.74 CKS1B (0.50) JAK1JAK2TYK2JAK3CKS1B
SCHEMBL28851424 0.74 JAK2 (0.44) JAK1JAK2TYK2JAK3KDM1A
SCHEMBL6942861 0.74 JAK2 (0.44) JAK1JAK2TYK2JAK3KDM1A
SCHEMBL6942857 0.74 JAK2 (0.44) JAK1JAK2TYK2JAK3KDM1A
SCHEMBL29062245 0.74 JAK2 (0.44) JAK1JAK2TYK2JAK3KDM1A
SCHEMBL28421562 0.74 BTK (0.38) JAK1JAK2TYK2JAK3KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111247119-B Amidine and guanidine derivatives, preparation method and application thereof in medicines 四川科伦博泰生物医药股份有限公司 2023-02-03 CN disclosed
CN-111247119-A Amidine and guanidine derivatives, preparation method and application thereof in medicines 四川科伦博泰生物医药股份有限公司 2020-06-05 CN disclosed