SCHEMBL28414964

SCHEMBL28414964

Cc1ccncc1C1CCC(NC(=O)OC(C)(C)C)CC1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 2/20 0.46
JAK1 P23458 4/20 0.46
JAK2 O60674 3/20 0.46
TYK2 P29597 1/20 0.46
JAK3 P52333 1/20 0.46
KDM1A O60341 1/20 0.46
MAOB P27338 1/20 0.46
KDM4D Q6B0I6 3/20 0.44
EPHX2 P34913 1/20 0.43
CKS1B P61024 1/20 0.42
SKP1 P63208 1/20 0.42
SKP2 Q13309 1/20 0.42
BTK Q06187 1/20 0.42
DRD2 P14416 3/20 0.41
CYP46A1 Q9Y6A2 1/20 0.41
SSTR4 P31391 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30209415 1.00 OPRL1 (0.46) OPRL1JAK1JAK2TYK2JAK3
SCHEMBL12326969 0.81 JAK1 (0.48) JAK1JAK2TYK2JAK3KDM1A
SCHEMBL28409256 0.79 JAK1 (0.50) JAK1JAK2TYK2JAK3KDM1A
SCHEMBL18795049 0.76 FDPS (0.43) KDM1AEPHX2
SCHEMBL15289131 0.76 KDM1A (0.44) JAK1JAK2KDM1AMAOBEPHX2
SCHEMBL9953027 0.75 GPR119 (0.43) SSTR4
SCHEMBL31206061 0.75 NAMPT (0.52) KDM1AMAOBEPHX2CKS1BSKP1
SCHEMBL3208745 0.75 ALDH1A1 (0.60) KDM1AMAOBEPHX2DRD2
SCHEMBL3208739 0.75 ALDH1A1 (0.60) KDM1AMAOBEPHX2DRD2
SCHEMBL6942861 0.75 JAK2 (0.44) JAK1JAK2TYK2JAK3KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111247119-B Amidine and guanidine derivatives, preparation method and application thereof in medicines 四川科伦博泰生物医药股份有限公司 2023-02-03 CN disclosed
CN-111247119-A Amidine and guanidine derivatives, preparation method and application thereof in medicines 四川科伦博泰生物医药股份有限公司 2020-06-05 CN disclosed