SCHEMBL28411531

SCHEMBL28411531

N#Cc1ccccc1-n1cc(-c2ccc(C=O)cc2)nn1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.45
ABCG2 Q9UNQ0 2/20 0.40
HSP90AA1 P07900 1/20 0.40
ABCB1 P08183 1/20 0.40
KDR P35968 3/20 0.38
MIF P14174 1/20 0.38
LDHA P00338 1/20 0.37
IRAK4 Q9NWZ3 1/20 0.36
MAPT P10636 1/20 0.36
KDM1A O60341 1/20 0.35
PTGS2 P35354 2/20 0.35
CA1 P00915 2/20 0.35
CA2 P00918 2/20 0.35
CA5A P35218 2/20 0.35
CA5B Q9Y2D0 2/20 0.35
CA12 O43570 1/20 0.35
CA9 Q16790 1/20 0.35
PTGS1 P23219 1/20 0.35
FLT3 P36888 1/20 0.35
GSK3B P49841 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28414389 0.80 BCHE (0.48) BCHEABCG2ABCB1KDRMIF
SCHEMBL28413622 0.80 BCHE (0.71) BCHEABCG2HSP90AA1ABCB1KDR
SCHEMBL28415505 0.80 FLT3 (0.56) BCHEABCG2ABCB1KDRMIF
SCHEMBL28410360 0.78 KDR (0.70) KDRMAPTFLT3GSK3B
SCHEMBL28410361 0.78 KDR (0.70) KDRMAPTFLT3GSK3B
SCHEMBL4549459 0.76 P2RX7 (0.58) BCHEKDRPTGS2CA1CA2
SCHEMBL28411507 0.76 CA1 (0.48) KDRPTGS2CA1CA2CA5A
SCHEMBL28414073 0.75 GRM5 (0.58) KDRCA1CA2CA12CA9
SCHEMBL29657622 0.75 GRM5 (0.58) KDRCA1CA2CA12CA9
SCHEMBL28335289 0.74 CA2 (0.61) BCHEKDRMIFPTGS2CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111153889-B 2-indolone-triazole anti-tumor compound and preparation method and application thereof 中国医科大学 2022-05-20 CN disclosed
CN-111153889-A 2-indolone-triazole anti-tumor compound and preparation method and application thereof 中国医科大学 2020-05-15 CN disclosed