SCHEMBL28413622

SCHEMBL28413622

O=Cc1ccc(-c2cn(-c3ccccc3Cl)nn2)cc1

nearest known ligand 0.71

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.71
TYMS P04818 3/20 0.48
NOTUM Q6P988 1/20 0.47
ABCG2 Q9UNQ0 2/20 0.42
ABCB1 P08183 1/20 0.42
KDR P35968 2/20 0.40
FLT3 P36888 2/20 0.40
GSK3B P49841 2/20 0.40
MIF P14174 1/20 0.40
LDHA P00338 1/20 0.39
PTGS2 P35354 4/20 0.39
PTGS1 P23219 2/20 0.39
CA2 P00918 2/20 0.38
CA5A P35218 2/20 0.38
CA9 Q16790 2/20 0.38
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA5B Q9Y2D0 1/20 0.37
HSP90AA1 P07900 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28046686 0.84 BCHE (1.00) BCHETYMSNOTUMABCG2ABCB1
SCHEMBL28414389 0.83 BCHE (0.48) BCHENOTUMABCG2ABCB1KDR
SCHEMBL28415505 0.83 FLT3 (0.56) BCHEABCG2ABCB1KDRFLT3
SCHEMBL28411531 0.80 BCHE (0.45) BCHEABCG2ABCB1KDRFLT3
SCHEMBL4549459 0.80 P2RX7 (0.58) BCHEKDRFLT3GSK3BPTGS2
SCHEMBL1230837 0.77 FLT3 (0.64) TYMSFLT3GSK3BPTGS2PTGS1
SCHEMBL28408386 0.77 FLT3 (0.69) TYMSNOTUMKDRFLT3GSK3B
SCHEMBL29657637 0.77 FLT3 (0.69) TYMSNOTUMKDRFLT3GSK3B
SCHEMBL28335289 0.77 CA2 (0.61) BCHEKDRFLT3GSK3BMIF
SCHEMBL28890847 0.76 KDR (0.74) BCHEKDRFLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111153889-B 2-indolone-triazole anti-tumor compound and preparation method and application thereof 中国医科大学 2022-05-20 CN disclosed
CN-111153889-A 2-indolone-triazole anti-tumor compound and preparation method and application thereof 中国医科大学 2020-05-15 CN disclosed