SCHEMBL28413196

SCHEMBL28413196

CC(NC(=O)c1cc(NC(=O)N2CCC(F)(F)CC2)ccc1N(C)C)c1ccccc1

nearest known ligand 0.66

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KCNB1 Q14721 3/20 0.66
KCNB2 Q92953 1/20 0.66
EPHX2 P34913 1/20 0.48
POLB P06746 2/20 0.42
KCNK3 O14649 2/20 0.41
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
LMNA P02545 1/20 0.41
HPGD P15428 1/20 0.41
HSD17B10 Q99714 1/20 0.41
NAMPT P43490 3/20 0.40
CNR1 P21554 1/20 0.40
CNR2 P34972 1/20 0.40
AURKA O14965 1/20 0.40
RPS6KB1 P23443 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
KCNH2 Q12809 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28402758 0.94 KCNB1 (0.63) KCNB1KCNB2EPHX2POLBKCNK3
SCHEMBL28402273 0.90 KCNB1 (0.60) KCNB1KCNB2EPHX2KDM4EALDH1A1
SCHEMBL28818685 0.89 KCNB1 (0.57) KCNB1KCNB2EPHX2POLBKCNK3
SCHEMBL28255850 0.81 KCNB1 (0.55) KCNB1KCNB2POLBKCNK3KDM4E
SCHEMBL29793705 0.80 KCNB1 (1.00) KCNB1KCNB2POLBKDM4EALDH1A1
SCHEMBL28255806 0.78 KCNB1 (0.53) KCNB1KCNB2POLBKCNK3KDM4E
SCHEMBL16583815 0.76 KCNB1 (0.69) KCNB1KCNB2POLBKCNK3LMNA
SCHEMBL28256075 0.75 KCNB1 (0.51) KCNB1KCNB2POLBKCNK3KDM4E
SCHEMBL27439889 0.72 ALDH1A1 (0.66) EPHX2POLBKDM4EALDH1A1HPGD
SCHEMBL28402250 0.72 KCNB1 (0.83) KCNB1KCNB2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108929263-B Arylamide Kv2.1 inhibitor and preparation method, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2022-07-22 CN disclosed
CN-111108092-A Arylamide Kv2.1 inhibitor and preparation method, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2020-05-05 CN disclosed