SCHEMBL28413640

SCHEMBL28413640

CNC(=O)c1ncccc1Oc1ccc(NC(=N)NC(=O)c2ccc(F)cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MET P08581 4/20 0.47
AXL P30530 4/20 0.47
MERTK Q12866 1/20 0.47
BRAF P15056 1/20 0.46
HDAC1 Q13547 1/20 0.46
KMT2A Q03164 2/20 0.44
RAB9A P51151 5/20 0.44
NPC1 O15118 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
LMNA P02545 1/20 0.44
KDR P35968 1/20 0.44
S1PR2 O95136 1/20 0.43
HIPK4 Q8NE63 1/20 0.43
F2 P00734 1/20 0.42
PLG P00747 1/20 0.42
PRSS1 P07477 1/20 0.42
PRSS2 P07478 1/20 0.42
PRSS3 P35030 1/20 0.42
ST14 Q9Y5Y6 1/20 0.42
MAPT P10636 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30448414 0.85 AXL (0.48) METAXLMERTKBRAFHDAC1
SCHEMBL28408407 0.82 KDM4E (0.39) METAXLMERTKBRAFHDAC1
SCHEMBL28850304 0.80 HIPK4 (0.64) METAXLMERTKBRAFHDAC1
SCHEMBL6049774 0.79 ALDH1A1 (0.46) BRAFHDAC1KMT2ARAB9ANPC1
SCHEMBL30448108 0.77 RAB9A (0.46) BRAFHDAC1KMT2ARAB9ANPC1
SCHEMBL30448073 0.76 KMT2A (0.51) BRAFHDAC1KMT2ARAB9ANPC1
SCHEMBL4265602 0.75 NAMPT (0.48) KMT2ARAB9ANPC1SMN1; SMN2LMNA
SCHEMBL4252286 0.74 MEN1 (0.45) BRAFHDAC1KMT2ASMN1; SMN2KDR
SCHEMBL29614703 0.74 MEN1 (0.45) BRAFHDAC1KMT2ASMN1; SMN2KDR
SCHEMBL5568329 0.71 RAF1 (0.64) METAXLMERTKBRAFKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107129465-B Aryl guanidine compound and preparation method and application thereof 中国科学院上海药物研究所 2020-06-19 CN disclosed