SCHEMBL28413656

SCHEMBL28413656

N#Cc1cc(-c2ccnc(Cl)n2)ncc1OC1CCC=CO1

nearest known ligand 0.36

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 2/20 0.36
TBK1 Q9UHD2 15/20 0.35
IKBKE Q14164 12/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20918320 0.79 TBK1 (0.52) TBK1IKBKE
SCHEMBL28890140 0.76 TBK1 (0.40) AAK1TBK1IKBKE
SCHEMBL1667272 0.65 TBK1 (0.64) TBK1IKBKE
SCHEMBL12448385 0.63 KMO (0.54) AAK1TBK1IKBKE
SCHEMBL14764257 0.62 IKBKE (0.56) AAK1TBK1IKBKE
SCHEMBL1667429 0.61 IKBKE (0.49) AAK1TBK1IKBKE
SCHEMBL1667504 0.61 KMO (0.49) AAK1TBK1IKBKE
SCHEMBL27881108 0.60 AAK1 (0.48) AAK1
SCHEMBL1667622 0.60 AAK1 (0.53) AAK1
SCHEMBL20929439 0.60 TBK1 (0.48) TBK1IKBKE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111247135-A Pyrimidine T-K/I-K-P inhibitor compound and application thereof 默克专利股份公司 2020-06-05 CN disclosed