SCHEMBL28416367

SCHEMBL28416367

O=Cc1ccc(-c2cn(-c3ccc(F)cc3)nn2)cc1

nearest known ligand 0.63

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 8/20 0.63
CA1 P00915 3/20 0.63
CA2 P00918 3/20 0.63
CA5A P35218 3/20 0.63
CA5B Q9Y2D0 3/20 0.63
PTGS1 P23219 3/20 0.63
FLT3 P36888 3/20 0.56
KDR P35968 2/20 0.50
CA12 O43570 2/20 0.50
CA9 Q16790 2/20 0.50
GSK3B P49841 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16220811 0.87 PTGS2 (0.72) PTGS2CA1CA2CA5ACA5B
SCHEMBL28418132 0.85 PTGS2 (0.64) PTGS2CA1CA2CA5ACA5B
SCHEMBL1230837 0.85 FLT3 (0.64) PTGS2CA1CA2CA5ACA5B
SCHEMBL28335289 0.85 CA2 (0.61) PTGS2CA1CA2CA5ACA5B
SCHEMBL4549459 0.85 P2RX7 (0.58) PTGS2CA1CA2CA5ACA5B
SCHEMBL28418357 0.83 STS (0.62) PTGS2CA1CA2CA5ACA5B
SCHEMBL29657629 0.83 STS (0.62) PTGS2CA1CA2CA5ACA5B
SCHEMBL28411507 0.82 CA1 (0.48) PTGS2CA1CA2CA5ACA5B
SCHEMBL18031100 0.80 PTGS2 (0.63) PTGS2CA1CA2CA5ACA5B
SCHEMBL23557718 0.80 PTGS2 (0.63) PTGS2CA1CA2CA5ACA5B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111153889-B 2-indolone-triazole anti-tumor compound and preparation method and application thereof 中国医科大学 2022-05-20 CN disclosed
CN-111153889-A 2-indolone-triazole anti-tumor compound and preparation method and application thereof 中国医科大学 2020-05-15 CN disclosed