SCHEMBL28416686

SCHEMBL28416686

NC(=O)OCCCN=C=O

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.39
CHRM2 P08172 2/20 0.38
CHRM4 P08173 2/20 0.38
CHRM5 P08912 2/20 0.38
CHRM1 P11229 2/20 0.38
CHRM3 P20309 2/20 0.38
CHRNB2 P17787 2/20 0.38
CHRNA4 P43681 2/20 0.38
HTR1A P08908 1/20 0.38
TSHR P16473 1/20 0.38
CYP2C19 P33261 1/20 0.38
CHRNA7 P36544 1/20 0.38
ALOX15 P16050 1/20 0.34
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
PRSS1 P07477 2/20 0.32
PRSS2 P07478 2/20 0.32
PRSS3 P35030 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22325445 0.92 PRSS1 (0.38) LMNACHRM2CHRM4CHRM5CHRM1
SCHEMBL16337241 0.87
SCHEMBL10481930 0.83 TSHR (0.31) TSHR
SCHEMBL9487597 0.79 ALDH1A1 (0.50) LMNACHRM2CHRM4CHRM5CHRM1
SCHEMBL8674490 0.79
Urethane SCHEMBL1054272 0.79 ALOX15 (0.56) LMNACHRM2CHRM4CHRM5CHRM1
SCHEMBL10482090 0.78 DGKA (0.44) TSHRPRSS1PRSS2PRSS3
Urethane SCHEMBL28162966 0.77 ALOX15 (0.54) LMNACHRM2TSHRALOX15PRSS1
SCHEMBL28405434 0.77 TSHR (0.45) LMNACHRM2CHRM4CHRM5CHRM1
SCHEMBL10481941 0.77 TSHR (0.34) TSHRPRSS1PRSS2PRSS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107660202-B Water-soluble prodrugs 大日本住友制药肿瘤公司 2021-12-24 CN disclosed
CN-111295368-A Chemically activated water soluble prodrugs 大日本住友制药株式会社 2020-06-16 CN disclosed