SCHEMBL28420192

SCHEMBL28420192

CC(C#CS)Cc1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 5/20 0.48
TAAR1 Q96RJ0 4/20 0.48
SLC6A2 P23975 3/20 0.48
SLC6A4 P31645 2/20 0.48
SLC6A3 Q01959 2/20 0.48
SIGMAR1 Q99720 2/20 0.48
CYP2A6 P11509 1/20 0.48
ADORA2A P29274 1/20 0.48
ADORA1 P30542 1/20 0.48
ADRA2B P18089 2/20 0.46
ADRA2C P18825 2/20 0.46
ADRA1A P35348 2/20 0.46
OPRK1 P41145 2/20 0.46
HTR2A P28223 1/20 0.46
KCNH2 Q12809 1/20 0.46
CYP2D6 P10635 3/20 0.45
SLC18A2 Q05940 1/20 0.45
MAOB P27338 6/20 0.44
CYP1A2 P05177 3/20 0.44
TSHR P16473 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19899811 0.81 SIGMAR1 (0.50) MAOATAAR1SLC6A2SLC6A4SLC6A3
SCHEMBL5594577 0.79 SIGMAR1 (0.48) MAOATAAR1SLC6A2SLC6A4SLC6A3
SCHEMBL367519 0.79 TRPA1 (0.48) MAOATAAR1SLC6A2SLC6A4SLC6A3
SCHEMBL3680285 0.78 TAAR1 (0.57) MAOATAAR1SLC6A2SLC6A4SLC6A3
SCHEMBL17802435 0.76 SIGMAR1 (0.50) MAOATAAR1SLC6A2SLC6A4SLC6A3
SCHEMBL2477572 0.76 SIGMAR1 (0.50) MAOATAAR1SLC6A2SLC6A4SLC6A3
SCHEMBL6387963 0.76 SIGMAR1 (0.54) MAOATAAR1SLC6A2SLC6A4SLC6A3
SCHEMBL8675172 0.74 SIGMAR1 (0.52) MAOATAAR1SLC6A2SLC6A4SLC6A3
SCHEMBL97558 0.74 TAAR1 (0.52) MAOATAAR1SLC6A2SLC6A4SLC6A3
SCHEMBL2748352 0.74 MAOB (0.56) MAOATAAR1SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111548299-A Preparation method of N-methyl-3-benzylmercapto-4-amino maleimide compound 温州医科大学 2020-08-18 CN claimed
CN-111393350-A Synthesis method of N-methyl-3-substituted benzylmercapto-4-morpholinyl maleimide compound 温州医科大学 2020-07-10 CN claimed
CN-111440108-A Synthetic method of N-substituted-3-benzylmercapto-4-morpholinyl maleimide compound 温州医科大学 2020-07-24 CN disclosed
CN-111440108-A Synthetic method of N-substituted-3-benzylmercapto-4-morpholinyl maleimide compound 温州医科大学 2020-07-24 CN disclosed
CN-111393350-A Synthesis method of N-methyl-3-substituted benzylmercapto-4-morpholinyl maleimide compound 温州医科大学 2020-07-10 CN disclosed