SCHEMBL28422136

SCHEMBL28422136

C[Si](C)(C)Oc1ccc(C=O)cc1F

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 11/20 0.47
TSHR P16473 1/20 0.47
HPGD P15428 2/20 0.44
MEN1 O00255 1/20 0.44
POLB P06746 1/20 0.44
KMT2A Q03164 1/20 0.44
AOX1 Q06278 1/20 0.43
GAA P10253 1/20 0.42
TUBB1 Q9H4B7 3/20 0.41
FDPS P14324 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
TRIM24 O15164 1/20 0.40
ALDH5A1 P51649 1/20 0.40
ABAT P80404 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
TRIM33 Q9UPN9 1/20 0.40
TTR P02766 1/20 0.38
MAPT P10636 2/20 0.36
KDM4E B2RXH2 1/20 0.36
BRD4 O60885 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3923554 0.83 ALDH1A1 (0.42) ALDH1A1TSHRHPGDMEN1POLB
SCHEMBL3673596 0.83 ALDH1A1 (0.57) ALDH1A1TSHRHPGDMEN1KMT2A
SCHEMBL30360257 0.83 ALDH1A1 (0.57) ALDH1A1TSHRHPGDMEN1KMT2A
SCHEMBL3689377 0.81 ALDH1A1 (0.43) ALDH1A1TSHRHPGDMEN1POLB
SCHEMBL7531959 0.79 ALDH1A1 (0.68) ALDH1A1TSHRHPGDMEN1POLB
SCHEMBL29400600 0.79 ALDH1A1 (0.68) ALDH1A1TSHRHPGDMEN1POLB
SCHEMBL435689 0.79 ALDH1A1 (0.68) ALDH1A1TSHRHPGDMEN1POLB
SCHEMBL9677313 0.79 ALDH1A1 (0.72) ALDH1A1TSHRHPGDMEN1KMT2A
SCHEMBL14033967 0.75 ALDH1A3 (0.52) ALDH1A1TSHRHPGDMEN1POLB
SCHEMBL2585951 0.75 ALDH1A1 (0.60) ALDH1A1TSHRHPGDMEN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111285874-A RET inhibitors, pharmaceutical compositions thereof and uses thereof 广东东阳光药业有限公司 2020-06-16 CN disclosed
CN-111285873-A RET inhibitors, pharmaceutical compositions thereof and uses thereof 广东东阳光药业有限公司 2020-06-16 CN disclosed