SCHEMBL28428697

SCHEMBL28428697

CCOC(=O)c1ccc2cc(F)ccc2n1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.64
CYP1A2 P05177 1/20 0.53
MAPT P10636 5/20 0.52
KDM4E B2RXH2 2/20 0.50
LMNA P02545 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
ALDH1A1 P00352 3/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
HPGD P15428 2/20 0.48
RAB9A P51151 2/20 0.48
NPC1 O15118 1/20 0.48
ALPL P05186 1/20 0.48
GAA P10253 1/20 0.48
GABRA2 P47869 1/20 0.47
GABRB2 P47870 1/20 0.47
PTPN1 P18031 1/20 0.44
HTR7 P34969 1/20 0.43
BACE1 P56817 1/20 0.42
TRPM8 Q7Z2W7 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8001647 0.85 CYP1A2 (0.56) TSHRCYP1A2MAPTKDM4ETDP1
SCHEMBL2210778 0.84 CYP1A2 (0.54) TSHRCYP1A2MAPTKDM4EALDH1A1
SCHEMBL14339761 0.83 MAPT (0.48) TSHRMAPTKDM4ELMNAALDH1A1
SCHEMBL1208379 0.82 CYP1A2 (0.53) TSHRCYP1A2MAPTKDM4ETDP1
SCHEMBL2001591 0.82 ALDH1A1 (0.65) TSHRCYP1A2MAPTKDM4ENPSR1
SCHEMBL28434347 0.81 KDM4E (0.65) CYP1A2MAPTKDM4ELMNANPSR1
SCHEMBL28231530 0.81 ALDH1A1 (0.48) TSHRCYP1A2MAPTKDM4EALDH1A1
SCHEMBL28428705 0.80 CYP1A2 (0.50) TSHRCYP1A2MAPTKDM4ELMNA
SCHEMBL1998568 0.79 CYP1A2 (0.49) TSHRCYP1A2MAPTKDM4ELMNA
SCHEMBL2002271 0.79 CYP1A2 (0.49) TSHRCYP1A2MAPTKDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108314647-B Preparation method of quinoline-2-formic acid and quinoline-2-formic acid derivative 华中科技大学 2020-06-26 CN claimed
CN-108314647-B Preparation method of quinoline-2-formic acid and quinoline-2-formic acid derivative 华中科技大学 2020-06-26 CN disclosed