SCHEMBL28429341

SCHEMBL28429341

c1csc(-c2ccc3c(c2)CCN3)n1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.45
DRD4 P21917 1/20 0.45
PDPK1 O15530 1/20 0.43
LOXL2 Q9Y4K0 1/20 0.42
PIK3CD O00329 1/20 0.40
S1PR1 P21453 2/20 0.40
ADRB2 P07550 1/20 0.40
S1PR3 Q99500 1/20 0.39
CYP2A6 P11509 1/20 0.39
CHEK1 O14757 1/20 0.38
JAK2 O60674 1/20 0.38
JAK3 P52333 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.36
SMPD3 Q9NY59 1/20 0.36
ABL1 P00519 1/20 0.35
BCR P11274 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
HDAC2 Q92769 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31164769 0.79 ASIC3 (0.55) DRD2PDPK1LOXL2
SCHEMBL28403784 0.77 DRD2 (0.63) DRD2DRD4PIK3CDS1PR1S1PR3
SCHEMBL29756191 0.77 DRD2 (0.63) DRD2DRD4PIK3CDS1PR1S1PR3
SCHEMBL9952071 0.76 DRD2 (0.42) DRD2DRD4PIK3CDS1PR1S1PR3
SCHEMBL27410695 0.76 PDPK1 (0.47) PDPK1LOXL2ADRB2CYP2A6CHEK1
SCHEMBL1459657 0.75 PDE3B (0.60) CHEK1
SCHEMBL8528347 0.74 DRD2 (0.47) DRD2DRD4PIK3CDS1PR1CYP2A6
SCHEMBL3874468 0.74 PDPK1 (0.46) PDPK1LOXL2ADRB2CYP2A6CHEK1
SCHEMBL20953202 0.74 DRD2 (0.38) DRD2DRD4PIK3CDS1PR1S1PR3
SCHEMBL2200009 0.73 SLC6A11 (0.47) DRD2DRD4S1PR1CYP2A6HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111471037-B Allylamine compound and application thereof 药捷安康(南京)科技股份有限公司 2023-02-10 CN disclosed
CN-111471037-A Allylamine compound and application thereof 南京药捷安康生物科技有限公司 2020-07-31 CN disclosed