SCHEMBL28430438

SCHEMBL28430438

COc1nc(Cl)c2ccc(OCc3ccccc3)cc2n1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.49
MAOB P27338 3/20 0.48
ALOX5 P09917 1/20 0.47
PDGFRB P09619 1/20 0.45
PDGFRA P16234 1/20 0.45
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
MAOA P21397 1/20 0.44
DHODH Q02127 1/20 0.42
KIT P10721 1/20 0.42
P2RY14 Q15391 1/20 0.42
ACHE P22303 1/20 0.41
IP6K1 Q92551 1/20 0.41
DYRK1A Q13627 1/20 0.41
MEN1 O00255 1/20 0.41
HSP90AA1 P07900 1/20 0.41
KMT2A Q03164 1/20 0.41
EGFR P00533 1/20 0.41
ERBB2 P04626 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4725521 0.90 MAOB (0.48) CYP3A4MAOBPDGFRBPDGFRADHODH
SCHEMBL856542 0.85 CYP3A4 (0.52) CYP3A4MAOBALOX5NPC1RAB9A
SCHEMBL28421218 0.85 CYP3A4 (0.49) CYP3A4MAOBALOX5PDGFRBPDGFRA
SCHEMBL6471210 0.81 EGFR (0.50) CYP3A4MAOBPDGFRBPDGFRANPC1
SCHEMBL13729181 0.80 ALDH1A1 (0.46) CYP3A4NPC1RAB9AACHEDYRK1A
SCHEMBL2329011 0.80 CYP3A4 (0.49) CYP3A4MAOBALOX5PDGFRBPDGFRA
SCHEMBL14931604 0.77 MAOB (0.54) MAOBMAOAACHEEGFR
SCHEMBL856483 0.77 CYP3A4 (0.51) CYP3A4MAOBALOX5NPC1RAB9A
SCHEMBL5033238 0.76 MAPT (0.54) CYP3A4MAOBALOX5NPC1RAB9A
SCHEMBL1012732 0.76 PIN1 (0.50) CYP3A4MAOBALOX5MAOAACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111253385-A Heterocyclic compound, preparation method and application 遵义医科大学珠海校区 2020-06-09 CN disclosed