SCHEMBL28430477

SCHEMBL28430477

O=C(O)COCCc1cn(CC(=O)O)c2ccccc12

nearest known ligand 0.60

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 5/20 0.60
ALDH1A1 P00352 3/20 0.51
TBXAS1 P24557 1/20 0.51
KMT2A Q03164 2/20 0.50
STAT3 P40763 1/20 0.50
KDM4E B2RXH2 3/20 0.48
PTGDR2 Q9Y5Y4 2/20 0.47
AKR1A1 P14550 1/20 0.47
AKR1B1 P15121 1/20 0.47
ALOX5 P09917 1/20 0.46
MAPT P10636 2/20 0.45
GFER P55789 1/20 0.45
GAA P10253 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8021536 0.81 MCL1 (0.60) MCL1ALDH1A1TBXAS1KMT2ASTAT3
SCHEMBL1520240 0.79 TBXAS1 (0.64) MCL1ALDH1A1TBXAS1KMT2ASTAT3
SCHEMBL28428521 0.79 ALDH1A1 (0.58) MCL1ALDH1A1KMT2AKDM4EALOX5
SCHEMBL18180209 0.78 CDC25A (0.63) MCL1ALDH1A1TBXAS1KMT2ASTAT3
SCHEMBL12874520 0.78 KMT2A (0.66) MCL1ALDH1A1TBXAS1KMT2ASTAT3
SCHEMBL6567317 0.77 ALDH1A1 (0.58) MCL1ALDH1A1TBXAS1KMT2ASTAT3
SCHEMBL9701519 0.76 KMT2A (0.60) ALDH1A1TBXAS1KMT2ASTAT3KDM4E
SCHEMBL16540887 0.75 MCL1 (1.00) MCL1PTGDR2
SCHEMBL8690315 0.74 S1PR2 (0.58) MCL1ALDH1A1TBXAS1KMT2ASTAT3
SCHEMBL30979650 0.73 ALDH1A1 (0.55) MCL1ALDH1A1TBXAS1KMT2ASTAT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109111501-B Fatty amino acid modified indole ethanol derivative, and synthesis, activity and application thereof 首都医科大学 2022-04-22 CN claimed
CN-109081801-B Acidic amino acid modified indoloethanol derivative, and synthesis, activity and application thereof 首都医科大学 2021-03-30 CN claimed
CN-109111390-B Met-modified indoloethanol derivative, and synthesis, activity and application thereof 首都医科大学 2021-03-30 CN claimed
CN-109081803-B Polar amino acid modified indoloethanol derivative, and synthesis, activity and application thereof 首都医科大学 2021-03-30 CN claimed
CN-109081802-B Indole ethanol derivative modified by basic amino acid, and synthesis, activity and application thereof 首都医科大学 2021-03-30 CN claimed
CN-108976159-B Aromatic amino acid modified indole ethanol derivative, and synthesis, activity and application thereof 首都医科大学 2020-07-28 CN claimed
CN-109111501-B Fatty amino acid modified indole ethanol derivative, and synthesis, activity and application thereof 首都医科大学 2022-04-22 CN disclosed
CN-109081801-B Acidic amino acid modified indoloethanol derivative, and synthesis, activity and application thereof 首都医科大学 2021-03-30 CN disclosed
CN-109081803-B Polar amino acid modified indoloethanol derivative, and synthesis, activity and application thereof 首都医科大学 2021-03-30 CN disclosed
CN-109111390-B Met-modified indoloethanol derivative, and synthesis, activity and application thereof 首都医科大学 2021-03-30 CN disclosed
CN-109081802-B Indole ethanol derivative modified by basic amino acid, and synthesis, activity and application thereof 首都医科大学 2021-03-30 CN disclosed
CN-108976159-B Aromatic amino acid modified indole ethanol derivative, and synthesis, activity and application thereof 首都医科大学 2020-07-28 CN disclosed