SCHEMBL28433786

SCHEMBL28433786

COc1ccc2nc(-c3ccccc3)c(=O)n(Cc3ccc(C(C)(C)C)cc3)c2c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CFTR P13569 5/20 0.55
CCR9 P51686 1/20 0.53
BRD4 O60885 1/20 0.53
TP53 P04637 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
USP2 O75604 4/20 0.50
ALDH1A1 P00352 4/20 0.50
CYP1A2 P05177 4/20 0.50
CYP3A4 P08684 4/20 0.50
CYP2C9 P11712 3/20 0.50
LMNA P02545 3/20 0.50
CYP2C19 P33261 3/20 0.50
HSD17B10 Q99714 3/20 0.50
CYP2D6 P10635 2/20 0.50
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
CASP1 P29466 2/20 0.48
CASP7 P55210 2/20 0.48
HPGD P15428 1/20 0.48
MAPK1 P28482 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29386548 1.00 CFTR (0.55) CFTRCCR9BRD4TP53SMN1; SMN2
SCHEMBL28430136 0.88 CFTR (0.57) CFTRBRD4USP2ALDH1A1CYP1A2
SCHEMBL29388744 0.88 CFTR (0.57) CFTRBRD4USP2ALDH1A1CYP1A2
SCHEMBL4311696 0.82 CCR9 (0.48) CFTRCCR9BRD4USP2ALDH1A1
SCHEMBL17184347 0.80 CFTR (0.59) CFTRBRD4TP53USP2ALDH1A1
SCHEMBL28430587 0.78 USP2 (0.49) CFTRBRD4TP53USP2ALDH1A1
SCHEMBL4659601 0.77 BRD4 (0.50) BRD4SMN1; SMN2ALDH1A1LMNAKMT2A
SCHEMBL4311048 0.77 SCD (0.51) BRD4USP2ALDH1A1CYP1A2CYP3A4
SCHEMBL28736739 0.75 ALDH1A1 (0.65) BRD4USP2ALDH1A1CYP1A2CYP3A4
SCHEMBL6475362 0.74 ALDH1A1 (0.74) BRD4TP53SMN1; SMN2ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111423388-B 7-methoxy-3-phenylquinoxaline-2 (1H) -one derivative and preparation method and application thereof 浙江工业大学 2022-02-15 CN disclosed
CN-111423388-A 7-methoxy-3-phenylquinoxaline-2 (1H) -one derivative and preparation method and application thereof 浙江工业大学 2020-07-17 CN disclosed