SCHEMBL28433865

SCHEMBL28433865

O=C(/C=C/c1ccccc1)NC(Cn1ccnc1)Cn1ccnc1

nearest known ligand 0.61

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.51
TBXAS1 P24557 4/20 0.50
CYP1A2 P05177 2/20 0.50
KMT2A Q03164 2/20 0.50
USP2 O75604 1/20 0.50
LMNA P02545 1/20 0.50
MEN1 O00255 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C19 P33261 1/20 0.50
TDP1 Q9NUW8 1/20 0.46
CYP19A1 P11511 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28433866 1.00 ALDH1A1 (0.51) ALDH1A1TBXAS1CYP1A2KMT2AUSP2
SCHEMBL28440838 0.88 ALDH1A1 (0.52) ALDH1A1TBXAS1CYP1A2KMT2AUSP2
SCHEMBL28433860 0.88 ALDH1A1 (0.52) ALDH1A1TBXAS1CYP1A2KMT2AUSP2
SCHEMBL28440915 0.85 TAS1R3 (0.61) ALDH1A1TBXAS1
SCHEMBL28442106 0.85 ALDH1A1 (0.49) ALDH1A1TBXAS1CYP1A2KMT2AUSP2
SCHEMBL28571346 0.81 TBXAS1 (0.47) TBXAS1CYP1A2KMT2AUSP2LMNA
SCHEMBL10858272 0.79 ALDH1A1 (0.79) ALDH1A1KMT2ALMNA
SCHEMBL10858265 0.79 ALDH1A1 (0.79) ALDH1A1KMT2ALMNA
SCHEMBL28450727 0.79 ALDH1A1 (0.40) ALDH1A1TBXAS1CYP1A2KMT2AUSP2
SCHEMBL28441964 0.78 KMT2A (0.53) ALDH1A1CYP1A2KMT2AMEN1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111533693-A Cinnamic acid amide diazole derivative and application thereof in antifungal drugs 张建蒙 2020-08-14 CN claimed
CN-111533693-A Cinnamic acid amide diazole derivative and application thereof in antifungal drugs 张建蒙 2020-08-14 CN disclosed