SCHEMBL28434603

SCHEMBL28434603

Cn1c(=O)c2c(-c3ccc(F)cc3)c(C(=O)c3ccc(F)cc3)nn2c2ccccc21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 2/20 0.45
GAA P10253 1/20 0.43
SMN1; SMN2 Q16637 3/20 0.40
MAPT P10636 3/20 0.40
LMNA P02545 2/20 0.40
TSHR P16473 1/20 0.40
MAPK1 P28482 1/20 0.40
AHR P35869 2/20 0.38
NPC1 O15118 3/20 0.38
RAB9A P51151 3/20 0.38
ALDH1A1 P00352 4/20 0.38
KDM4E B2RXH2 3/20 0.38
TDP1 Q9NUW8 2/20 0.38
TP53 P04637 1/20 0.38
POLB P06746 1/20 0.38
THRB P10828 1/20 0.38
PKM P14618 1/20 0.38
BLM P54132 1/20 0.38
CTDSP1 Q9GZU7 1/20 0.38
KMT2A Q03164 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28426049 0.88 KMT2A (0.43) GAASMN1; SMN2MAPTLMNAALDH1A1
SCHEMBL28430288 0.85 ADORA3 (0.41) SMN1; SMN2MAPTLMNATSHRMAPK1
SCHEMBL28428820 0.84 PADI4 (0.45) GAASMN1; SMN2LMNAAHRALDH1A1
SCHEMBL28430717 0.82 POLB (0.46) SMN1; SMN2MAPTLMNAMAPK1NPC1
SCHEMBL28431825 0.76 SMN1; SMN2 (0.46) MAPK14GAASMN1; SMN2MAPTLMNA
SCHEMBL28438083 0.72 RAB9A (0.59) GAASMN1; SMN2MAPTLMNATSHR
SCHEMBL4203809 0.70 MEN1 (0.61) SMN1; SMN2MAPTLMNANPC1RAB9A
SCHEMBL28428727 0.68 ADORA3 (0.42) MAPK14SMN1; SMN2MAPTLMNATSHR
SCHEMBL4200653 0.68 SMN1; SMN2 (0.54) SMN1; SMN2MAPTLMNATSHRALDH1A1
SCHEMBL24864974 0.65 KMT2A (0.66) GAASMN1; SMN2MAPTLMNANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108148064-B Method for preparing pyrazole quinoxalinone derivative 浙江百斯特化工有限公司 2020-06-26 CN disclosed