SCHEMBL28434682

SCHEMBL28434682

CN(C)Cc1nc2ccc([N+](=O)[O-])cc2[nH]1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.69
ALDH1A1 P00352 5/20 0.68
MAPT P10636 5/20 0.68
KCNJ1 P48048 2/20 0.68
LMNA P02545 1/20 0.68
RIPK1 Q13546 4/20 0.62
PKM P14618 2/20 0.62
TDP1 Q9NUW8 2/20 0.57
SMN1; SMN2 Q16637 4/20 0.57
L3MBTL1 Q9Y468 2/20 0.57
HPGD P15428 1/20 0.55
NPC1 O15118 4/20 0.55
RAB9A P51151 4/20 0.55
HTT P42858 3/20 0.55
MMP2 P08253 1/20 0.55
MMP9 P14780 1/20 0.55
MMP8 P22894 1/20 0.55
CASP3 P42574 1/20 0.55
MMP13 P45452 1/20 0.55
SENP8 Q96LD8 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28439013 0.86 KDM4E (0.70) KDM4EALDH1A1MAPTKCNJ1LMNA
SCHEMBL28432878 0.85 KDM4E (0.64) KDM4EALDH1A1MAPTKCNJ1LMNA
SCHEMBL6753969 0.84 KDM4E (0.79) KDM4EALDH1A1MAPTKCNJ1LMNA
SCHEMBL18459774 0.82 MAPT (0.76) KDM4EALDH1A1MAPTKCNJ1LMNA
SCHEMBL8601357 0.82 KDM4E (1.00) KDM4EALDH1A1MAPTKCNJ1LMNA
SCHEMBL18426060 0.81 MAPT (0.74) KDM4EALDH1A1MAPTKCNJ1LMNA
SCHEMBL9642133 0.81 MAPT (1.00) KDM4EALDH1A1MAPTKCNJ1LMNA
SCHEMBL16061454 0.81 MAPT (0.74) KDM4EALDH1A1MAPTKCNJ1LMNA
SCHEMBL1539990 0.81 ALDH1A1 (0.74) KDM4EALDH1A1MAPTKCNJ1LMNA
SCHEMBL521103 0.81 PKM (0.75) KDM4EALDH1A1MAPTKCNJ1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111484484-B 2, 4-diaryl aminopyrimidine derivative containing aromatic heterocycle and preparation and application thereof 沈阳药科大学 2021-11-23 CN disclosed
CN-111484484-A 2, 4-diaryl aminopyrimidine derivative containing aromatic heterocycle and preparation and application thereof 沈阳药科大学 2020-08-04 CN disclosed