SCHEMBL28439711

SCHEMBL28439711

CCCOc1c(Cl)ccc2c1OCC=C2

nearest known ligand 0.32

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.32
CSNK2A1 P68400 2/20 0.31
HTR2C P28335 2/20 0.30
HTR2B P41595 2/20 0.30
CYP1A1 P04798 1/20 0.30
CYP1A2 P05177 1/20 0.30
MAPT P10636 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28445516 0.75 CYP1A1 (0.32) CYP1A1CYP1A2
SCHEMBL28445561 0.74 CYP2A6 (0.41) HTR2CHTR2BNPSR1
SCHEMBL28441377 0.71 CYP1A1 (0.32) CYP1A1CYP1A2
SCHEMBL93424 0.70 AHR (0.38) KDM4ECSNK2A1MAPTNPSR1
SCHEMBL17826761 0.65 L3MBTL1 (0.56) KDM4ECSNK2A1MAPT
SCHEMBL28443125 0.63 KCNH2 (0.32)
SCHEMBL19122260 0.63 KDM4E (0.42) KDM4ECSNK2A1CYP1A2MAPT
SCHEMBL30629208 0.62 CYP2B6 (0.38) CYP1A1CYP1A2
SCHEMBL30623113 0.61 KDM4E (0.42) KDM4ECYP1A1CYP1A2MAPT
SCHEMBL1477385 0.60 CA1 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111417396-A Methods of treating cancer with small molecule NF-kB inhibitors 免疫目标公司 2020-07-14 CN disclosed