SCHEMBL28440209

SCHEMBL28440209

O=C(CCCc1cc(F)c(F)cc1F)N1CCCC1

nearest known ligand 0.59

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.52
ALDH1A1 P00352 1/20 0.48
DPP4 P27487 2/20 0.45
TRPV1 Q8NER1 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
NPC1 O15118 1/20 0.44
TDP1 Q9NUW8 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24725614 0.98 ATM (0.50) ATMALDH1A1DPP4TRPV1L3MBTL1
SCHEMBL23272135 0.78 DPP4 (0.55) DPP4L3MBTL1TDP1
SCHEMBL28435927 0.75 DPP4 (0.45) DPP4
SCHEMBL7891864 0.75 DPP4 (0.67) DPP4
SCHEMBL30427892 0.74 F13A1 (0.50)
SCHEMBL536350 0.74 F13A1 (0.50)
SCHEMBL25840260 0.74 DPP4 (0.44) DPP4
SCHEMBL5001351 0.73 NPC1 (0.57) NPC1TDP1
SCHEMBL8092673 0.72 NPC1 (0.55) TRPV1NPC1TDP1
SCHEMBL13501505 0.72 DPP4 (0.40) DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111534494-B (R) -omega-transaminase mutant and application thereof in preparation of sitagliptin intermediate 浙江工业大学 2021-10-01 CN claimed
CN-111411095-B Recombinant (R) -omega-transaminase, mutant and application thereof 浙江工业大学 2021-07-23 CN claimed
CN-111534494-A (R) -omega-transaminase mutant and application thereof in preparation of sitagliptin intermediate 浙江工业大学 2020-08-14 CN claimed
CN-111411095-A Novel recombinant (R) -omega-transaminase, mutant and application thereof 浙江工业大学 2020-07-14 CN claimed
CN-111534494-B (R) -omega-transaminase mutant and application thereof in preparation of sitagliptin intermediate 浙江工业大学 2021-10-01 CN disclosed
CN-111534494-B (R) -omega-transaminase mutant and application thereof in preparation of sitagliptin intermediate 浙江工业大学 2021-10-01 CN disclosed
CN-111411095-B Recombinant (R) -omega-transaminase, mutant and application thereof 浙江工业大学 2021-07-23 CN disclosed
CN-111534494-A (R) -omega-transaminase mutant and application thereof in preparation of sitagliptin intermediate 浙江工业大学 2020-08-14 CN disclosed
CN-111534494-A (R) -omega-transaminase mutant and application thereof in preparation of sitagliptin intermediate 浙江工业大学 2020-08-14 CN disclosed
CN-111411095-A Novel recombinant (R) -omega-transaminase, mutant and application thereof 浙江工业大学 2020-07-14 CN disclosed