SCHEMBL28440693

SCHEMBL28440693

O=C(O)c1cncc(Cl)c1O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C2 P52895 6/20 0.52
AKR1C1 Q04828 6/20 0.52
AKR1C4 P17516 1/20 0.52
AKR1C3 P42330 1/20 0.52
HCAR2 Q8TDS4 1/20 0.42
ALDH1A1 P00352 6/20 0.41
TTR P02766 1/20 0.41
HSD17B10 Q99714 3/20 0.41
KDM4E B2RXH2 3/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
HPGD P15428 2/20 0.41
MAPT P10636 2/20 0.41
PKM P14618 1/20 0.41
HTT P42858 1/20 0.41
DPP4 P27487 1/20 0.40
TSHR P16473 3/20 0.39
RXFP1 Q9HBX9 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
TP53 P04637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20512962 0.85 SELL (0.42) AKR1C2AKR1C1AKR1C4AKR1C3HCAR2
SCHEMBL392397 0.82 TSHR (0.48) AKR1C2AKR1C1AKR1C4AKR1C3HCAR2
SCHEMBL7067360 0.81 SELL (0.50) ALDH1A1HSD17B10KDM4EMEN1KMT2A
SCHEMBL29157397 0.78 HCAR2 (0.39) AKR1C2AKR1C1AKR1C4AKR1C3HCAR2
SCHEMBL535543 0.78 HAVCR2 (0.47) AKR1C2AKR1C1AKR1C4AKR1C3HCAR2
SCHEMBL15758062 0.78 HCAR2 (0.46) AKR1C2AKR1C1AKR1C4AKR1C3HCAR2
SCHEMBL2681685 0.77
SCHEMBL15334246 0.76 AKR1C3 (0.50) AKR1C2AKR1C1AKR1C4AKR1C3HCAR2
SCHEMBL31538840 0.76 KDM4E (0.53) HCAR2ALDH1A1HSD17B10KDM4EMEN1
SCHEMBL9311927 0.76 KDM4E (0.50) HCAR2ALDH1A1HSD17B10KDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110483388-B Preparation method of nicotinic acid derivative 新发药业有限公司 2020-08-04 CN disclosed
CN-110483388-B Preparation method of nicotinic acid derivative 新发药业有限公司 2020-08-04 CN disclosed