SCHEMBL29157397

SCHEMBL29157397

O=C(O)c1cncc(Cl)c1Br

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 3/20 0.39
POLB P06746 1/20 0.39
ALDH1A1 P00352 4/20 0.39
TSHR P16473 3/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
TP53 P04637 1/20 0.36
CASP1 P29466 1/20 0.36
AKR1C4 P17516 1/20 0.35
AKR1C3 P42330 1/20 0.35
AKR1C2 P52895 1/20 0.35
AKR1C1 Q04828 1/20 0.35
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
KDM6B O15054 1/20 0.34
KDM4A O75164 1/20 0.34
MAPT P10636 1/20 0.34
THRB P10828 1/20 0.34
KMT2A Q03164 1/20 0.34
KDM4D Q6B0I6 1/20 0.34
KDM4C Q9H3R0 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20111331 0.84 HCAR2 (0.46) HCAR2POLBALDH1A1TSHRAKR1C4
SCHEMBL28440693 0.78 AKR1C2 (0.52) HCAR2ALDH1A1TSHRSMN1; SMN2TP53
SCHEMBL392397 0.78 TSHR (0.48) HCAR2ALDH1A1TSHRSMN1; SMN2TP53
SCHEMBL659061 0.78 HCAR2 (0.42) HCAR2POLBALDH1A1TSHRAKR1C4
SCHEMBL3720517 0.75 HCAR2 (0.39) HCAR2POLBALDH1A1TSHRSMN1; SMN2
SCHEMBL31450301 0.75 HCAR2 (0.39) HCAR2POLBALDH1A1TSHRSMN1; SMN2
SCHEMBL12164567 0.75 HCAR2 (0.39) HCAR2POLBALDH1A1TSHRAKR1C4
SCHEMBL535543 0.75 HAVCR2 (0.47) HCAR2POLBALDH1A1TSHRSMN1; SMN2
SCHEMBL15758062 0.75 HCAR2 (0.46) HCAR2POLBALDH1A1TSHRSMN1; SMN2
SCHEMBL7905113 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117263853-A Method for synthesizing 4-bromo-5-chloro-nicotinic acid in one step 常州中氪生命科学技术有限公司 2023-12-22 CN claimed
CN-117263853-A Method for synthesizing 4-bromo-5-chloro-nicotinic acid in one step 常州中氪生命科学技术有限公司 2023-12-22 CN disclosed
CN-117263853-A Method for synthesizing 4-bromo-5-chloro-nicotinic acid in one step 常州中氪生命科学技术有限公司 2023-12-22 CN disclosed
CN-117263853-A Method for synthesizing 4-bromo-5-chloro-nicotinic acid in one step 常州中氪生命科学技术有限公司 2023-12-22 CN disclosed