SCHEMBL28440775

SCHEMBL28440775

CCCC1CNCCC1(c1cc[c]cc1)c1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 4/20 0.36
SLC6A9 P48067 2/20 0.36
HTR2A P28223 2/20 0.33
ADRB2 P07550 1/20 0.30
HTR1A P08908 1/20 0.30
SLC6A2 P23975 1/20 0.30
SLC6A4 P31645 1/20 0.30
ADRA1A P35348 1/20 0.30
HTR2B P41595 1/20 0.30
SLC6A3 Q01959 1/20 0.30
TACR1 P25103 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7216822 0.75 OPRM1 (0.39) OPRM1HTR2AHTR2BTACR1
SCHEMBL8642209 0.75 HTR2A (0.38) OPRM1HTR2AHTR1ASLC6A2SLC6A4
SCHEMBL7237713 0.69 KIF11 (0.40) OPRM1TACR1
SCHEMBL28536576 0.68 KDM4E (0.40) OPRM1HTR2ASLC6A2SLC6A4TACR1
SCHEMBL8642204 0.64 OPRM1 (0.36) OPRM1HTR2ASLC6A4TACR1
SCHEMBL30352945 0.63 ARG1 (0.31)
SCHEMBL29290911 0.62 OPRM1 (0.43) OPRM1HTR2ATACR1
SCHEMBL6847573 0.62 OPRM1 (0.37) OPRM1HTR2A
SCHEMBL11471276 0.62 OPRM1 (0.40) OPRM1HTR2ATACR1
SCHEMBL11451165 0.62 OPRM1 (0.40) OPRM1HTR2ATACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107074816-B Heterocyclic derivative, preparation method and medical application thereof 四川海思科制药有限公司 2020-07-17 CN disclosed