SCHEMBL28444583

SCHEMBL28444583

O=C(O)CCNC(=O)c1cc(Br)ccc1[N+](=O)[O-]

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
APEX1 P27695 1/20 0.48
ALDH1A1 P00352 4/20 0.43
HPGD P15428 2/20 0.43
MAPT P10636 1/20 0.43
AKR1C2 P52895 1/20 0.43
AKR1C1 Q04828 1/20 0.43
LMNA P02545 2/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
SIRT5 Q9NXA8 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
KDM4E B2RXH2 1/20 0.40
SIRT6 Q8N6T7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21296309 0.80 HPGD (0.63) HPGDNPC1RAB9ASMN1; SMN2CYP1A2
SCHEMBL18130511 0.77 PKM (0.46) ALDH1A1HPGDMAPTAKR1C2AKR1C1
SCHEMBL9335696 0.77 LMNA (0.47) ALDH1A1HPGDMAPTLMNANPC1
SCHEMBL7447850 0.77 SLC6A2 (0.48) ALDH1A1AKR1C2AKR1C1RAB9ASMN1; SMN2
SCHEMBL30566926 0.76 DTYMK (0.62) APEX1ALDH1A1AKR1C2AKR1C1LMNA
SCHEMBL1228589 0.76 DTYMK (0.62) APEX1ALDH1A1AKR1C2AKR1C1LMNA
SCHEMBL15206115 0.75 APEX1 (0.61) APEX1ALDH1A1HPGDMAPTNPC1
SCHEMBL13025484 0.74 DTYMK (0.56) ALDH1A1HPGDMAPTLMNASIRT5
SCHEMBL9336044 0.74 SIRT5 (0.39) ALDH1A1HPGDMAPTNPC1RAB9A
SCHEMBL10489202 0.73 HPGD (0.58) ALDH1A1HPGDMAPTLMNANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107428754-B Bicyclic quinazolinone derivatives 豪夫迈·罗氏有限公司 2020-07-31 CN disclosed