SCHEMBL28445347

SCHEMBL28445347

COC(=O)CCc1c[nH]c2cc(Br)ccc12

nearest known ligand 0.60

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.60
CHRNA7 P36544 1/20 0.60
CHRNA4 P43681 1/20 0.60
NPC1 O15118 1/20 0.52
MTNR1A P48039 3/20 0.51
MTNR1B P49286 3/20 0.51
EGFR P00533 1/20 0.50
MEN1 O00255 4/20 0.49
KMT2A Q03164 4/20 0.49
MAPT P10636 2/20 0.49
CDK2 P24941 3/20 0.47
NR4A2 P43354 1/20 0.47
HTR2A P28223 2/20 0.44
POLB P06746 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
TRPM8 Q7Z2W7 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3030323 0.89 MTNR1A (0.64) MTNR1AMTNR1BMEN1KMT2AMAPT
SCHEMBL498040 0.86 CHRNB2 (0.56) CHRNB2CHRNA7CHRNA4NPC1MTNR1A
SCHEMBL29506986 0.86 CHRNB2 (0.56) CHRNB2CHRNA7CHRNA4NPC1MTNR1A
SCHEMBL15323543 0.85 HTR2C (0.58) NPC1MTNR1AMTNR1BMEN1KMT2A
SCHEMBL20931043 0.84 HPGD (0.56) NPC1MTNR1AMTNR1BMEN1KMT2A
SCHEMBL30517178 0.83 CHRNB2 (0.58) CHRNB2CHRNA7CHRNA4NPC1MTNR1A
SCHEMBL7423854 0.83 NPC1 (0.76) NPC1MTNR1AMTNR1BMEN1KMT2A
SCHEMBL24448409 0.81 CDK2 (0.50) NPC1MTNR1AMTNR1BMEN1KMT2A
SCHEMBL4605682 0.81 MTNR1A (0.55) NPC1MTNR1AMTNR1BMEN1KMT2A
Methyl 3-(3-Indolylmethyl)Propanoate SCHEMBL290808 0.80 MAPT (0.71) MEN1KMT2AMAPTPOLBTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111499591-A ROR gamma modulators 山东轩竹医药科技有限公司 2020-08-07 CN disclosed