SCHEMBL28445360

SCHEMBL28445360

CCOC(=O)C[C@@H](C)Cc1ccc(Cl)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.48
EPHX2 P34913 1/20 0.46
PPARG P37231 3/20 0.43
PPARA Q07869 3/20 0.43
SLC6A2 P23975 1/20 0.43
SLC6A3 Q01959 1/20 0.43
ALDH1A1 P00352 4/20 0.43
KDM4E B2RXH2 2/20 0.43
LMNA P02545 2/20 0.43
NPSR1 Q6W5P4 2/20 0.43
TNF P01375 1/20 0.43
HSP90AA1 P07900 1/20 0.43
HPGD P15428 1/20 0.43
ALOX12 P18054 1/20 0.43
CCR6 P51684 1/20 0.43
RUNX1 Q01196 1/20 0.43
CBFB Q13951 1/20 0.43
HKDC1 Q2TB90 1/20 0.43
NOD2 Q9HC29 1/20 0.43
GPR35 Q9HC97 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2303859 0.86 ESR1 (0.46) SLC6A2KMT2A
SCHEMBL27481292 0.85 HDAC3 (0.47) MAPTEPHX2PPARGPPARASLC6A2
SCHEMBL12446348 0.84 MMP8 (0.51) ALDH1A1LMNAMEN1KMT2ATSHR
SCHEMBL2431295 0.83 LDHA (0.53) MAPTEPHX2ALDH1A1KDM4ELMNA
SCHEMBL17335899 0.83 SLC6A4 (0.53) MAPTEPHX2PPARGPPARASLC6A2
SCHEMBL14741319 0.82 PNMT (0.50) MAPTPPARGPPARAALDH1A1KDM4E
SCHEMBL8362177 0.81 MAPT (0.48) MAPTEPHX2PPARGPPARAALDH1A1
SCHEMBL11835523 0.81 TSHR (0.45) MAPTEPHX2PPARGPPARAALDH1A1
SCHEMBL11357662 0.80 CTSC (0.45) MAPTEPHX2PPARGPPARAALDH1A1
SCHEMBL27884796 0.79 PPARG (0.47) MAPTEPHX2PPARGPPARAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111587238-A Manganese catalyzed ester hydrogenation 圣安德鲁斯大学董事会 2020-08-25 CN disclosed