SCHEMBL28447697

SCHEMBL28447697

Nc1ccnc(-c2cnc(C(F)(F)F)nc2)n1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.38
NOS2 P35228 1/20 0.38
ALOX5AP P20292 6/20 0.37
FEN1 P39748 6/20 0.37
IRAK4 Q9NWZ3 1/20 0.35
KCNH2 Q12809 1/20 0.35
SCN9A Q15858 1/20 0.35
S1PR1 P21453 2/20 0.34
DHFR P00374 1/20 0.34
S1PR3 Q99500 1/20 0.34
PIK3CD O00329 1/20 0.33
IDO1 P14902 1/20 0.33
FGFR3 P22607 1/20 0.33
KDR P35968 1/20 0.33
TRPV3 Q8NET8 1/20 0.33
HDAC4 P56524 1/20 0.33
MET P08581 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3794168 0.77 TRPV3 (0.48) NOS3NOS2KCNH2SCN9AS1PR1
SCHEMBL17609513 0.76 IRAK4 (0.39) NOS3NOS2ALOX5APFEN1IRAK4
SCHEMBL19066984 0.76 NOS3 (0.50) NOS3NOS2ALOX5APFEN1KCNH2
SCHEMBL17609652 0.75 S1PR1 (0.43) NOS3NOS2ALOX5APFEN1IRAK4
SCHEMBL1420222 0.75 NOS3 (0.47) NOS3NOS2ALOX5APFEN1KCNH2
SCHEMBL28898005 0.75 CYP2A6 (0.40) DHFRHDAC4
SCHEMBL30462066 0.74 HSP90AA1 (0.40) ALOX5APFEN1IRAK4
SCHEMBL30911587 0.74 CYP2A6 (0.40) ALOX5APFEN1IRAK4KDR
SCHEMBL17609846 0.72 ASIC3 (0.52) NOS3NOS2IRAK4DHFRPIK3CD
SCHEMBL18018441 0.72 KDR (0.36) DHFRPIK3CDFGFR3KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107922392-B 1- (hetero) arylsulfonyl- (pyrrolidine or piperidine) -2-carboxamide derivatives and uses thereof 豪夫迈·罗氏有限公司 2020-07-21 CN disclosed