SCHEMBL28447997

SCHEMBL28447997

NC(=O)OC1CCN(c2cccnc2)CC1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 1/20 0.53
AOC3 Q16853 3/20 0.47
CHRNB2 P17787 5/20 0.46
CHRNA4 P43681 5/20 0.46
CHRNB4 P30926 2/20 0.46
CHRNA3 P32297 2/20 0.46
HRH3 Q9Y5N1 2/20 0.45
DPP4 P27487 2/20 0.44
DPP8 Q6V1X1 2/20 0.44
DPP9 Q86TI2 2/20 0.44
DPP7 Q9UHL4 2/20 0.44
NPY5R Q15761 1/20 0.43
FFAR1 O14842 1/20 0.43
TRPV6 Q9H1D0 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28379144 0.82 POLB (0.52) GPR119HRH3
SCHEMBL16684777 0.82 HRH3 (0.43) AOC3HRH3
SCHEMBL4392645 0.81 GPR119 (0.53) GPR119AOC3CHRNB2CHRNA4CHRNB4
SCHEMBL30663949 0.81 GPR119 (0.53) GPR119AOC3CHRNB2CHRNA4CHRNB4
SCHEMBL21828535 0.81 GPR119 (0.51) GPR119CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL28719495 0.80 HRH3 (0.51) GPR119AOC3CHRNB2CHRNA4CHRNB4
SCHEMBL27600357 0.78 CHRNB2 (0.51) GPR119CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL19302597 0.78 GPR119 (0.52) GPR119CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL31329886 0.78 GPR119 (0.52) GPR119CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL20483697 0.78 HRH3 (0.50) HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107629059-B Compounds useful as inhibitors of ATR kinase 沃泰克斯药物股份有限公司 2020-07-28 CN disclosed