SCHEMBL2844811

SCHEMBL2844811

CC(=O)N(CCOC(=O)Nc1ccc(C(F)(F)F)cn1)NCc1ccccc1Cl.CC(=O)N(CCON(C=O)c1ccc(C#N)cn1)NCc1ccccc1Cl

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 2/20 0.33
CNR2 P34972 2/20 0.33
DYRK3 O43781 1/20 0.32
GSK3A P49840 1/20 0.32
GSK3B P49841 1/20 0.32
DYRK1A Q13627 1/20 0.32
CLK4 Q9HAZ1 1/20 0.32
STK17A Q9UEE5 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
RPS6KA3 P51812 1/20 0.32
NPSR1 Q6W5P4 1/20 0.31
HCRTR1 O43613 1/20 0.31
VNN1 O95497 1/20 0.31
POLB P06746 1/20 0.31
GAA P10253 1/20 0.31
CHEK1 O14757 1/20 0.30
CYP3A4 P08684 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4343021 0.97 CNR1 (0.31) CNR1CNR2DYRK3GSK3AGSK3B
SCHEMBL15808665 0.87 CNR1 (0.33) CNR1CNR2DYRK3GSK3AGSK3B
SCHEMBL209728 0.86 EPHX2 (0.37) RPS6KA3NPSR1HCRTR1POLBGAA
SCHEMBL210066 0.86 VNN1 (0.39) VNN1CHEK1CYP3A4
SCHEMBL15808659 0.79
SCHEMBL210702 0.76 NR3C1 (0.38) NPC1RAB9APOLBCYP3A4
SCHEMBL14719091 0.76 NPC1 (0.34) NPC1RAB9A
SCHEMBL213609 0.76 P2RX7 (0.35) NPC1RAB9ACYP3A4
SCHEMBL212585 0.74 HTT (0.35) NPSR1
SCHEMBL210503 0.74 EPHX2 (0.33) NPC1RAB9ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2195328-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS Cytokinetics, Incorporated (US) 2010-06-16 EP disclosed
WO-2009023193-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INCORPORATED (US) 2009-02-19 WO disclosed